SCHEMBL2851391

SCHEMBL2851391

Cc1ccc(C(=O)N[C@@H]2CON(CCO)C2=O)cc1-n1cnc(OCc2ccc(F)cc2F)c(Cl)c1=O

nearest known ligand 0.69

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 20/20 0.69
MAPK11 Q15759 4/20 0.69
ROCK2 O75116 1/20 0.43
MAPK12 P53778 1/20 0.43
STRADA Q7RTN6 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2851394 1.00 MAPK14 (0.69) MAPK14MAPK11ROCK2MAPK12STRADA
SCHEMBL2847861 0.94 MAPK14 (0.64) MAPK14MAPK11ROCK2MAPK12STRADA
SCHEMBL9906477 0.94 MAPK14 (0.64) MAPK14MAPK11ROCK2MAPK12STRADA
SCHEMBL2847864 0.94 MAPK14 (0.64) MAPK14MAPK11ROCK2MAPK12STRADA
SCHEMBL2851673 0.92 MAPK14 (0.68) MAPK14MAPK11ROCK2MAPK12STRADA
SCHEMBL2851670 0.92 MAPK14 (0.68) MAPK14MAPK11ROCK2MAPK12STRADA
SCHEMBL2851949 0.87 MAPK14 (0.70) MAPK14MAPK11ROCK2MAPK12STRADA
SCHEMBL2851945 0.87 MAPK14 (0.70) MAPK14MAPK11ROCK2MAPK12STRADA
SCHEMBL13287648 0.87 MAPK14 (0.70) MAPK14MAPK11ROCK2MAPK12STRADA
SCHEMBL2849958 0.86 MAPK14 (0.62) MAPK14MAPK11ROCK2MAPK12STRADA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8198276-B2 Kinase inhibitor compounds XCOVERY HOLDING COMPANY LLC (US) 2012-06-12 US disclosed
US-8198276-B2 Kinase inhibitor compounds XCOVERY HOLDING COMPANY LLC (US) 2012-06-12 US disclosed
US-8198276-B2 Kinase inhibitor compounds XCOVERY HOLDING COMPANY LLC (US) 2012-06-12 US disclosed
US-20100144768-A1 KINASE INHIBITOR COMPOUNDS COMPASS HORIZON FUNDING COMPANY LLC 2010-06-10 US disclosed
US-20100144768-A1 KINASE INHIBITOR COMPOUNDS COMPASS HORIZON FUNDING COMPANY LLC 2010-06-10 US disclosed
US-20100144768-A1 KINASE INHIBITOR COMPOUNDS COMPASS HORIZON FUNDING COMPANY LLC 2010-06-10 US disclosed
EP-2166857-A1 KINASE INHIBITOR COMPOUNDS Xcovery, INC. (US) 2010-03-31 EP disclosed
WO-2008153942-A1 KINASE INHIBITOR COMPOUNDS XCOVERY, INC. (US) 2008-12-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100144768-A1 KINASE INHIBITOR COMPOUNDS MAP3K9, MAP3K1, MAP3K8 MAPK14 183/4885MAPK11 413/4885ROCK2 557/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.