SCHEMBL28515229

SCHEMBL28515229

Nc1cc(Oc2ccc(F)cc2F)c(Br)cn1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EPAS1 Q99814 1/20 0.44
MAPK14 Q16539 1/20 0.43
MAP4K4 O95819 1/20 0.42
TRPA1 O75762 13/20 0.41
HSPB1 P04792 1/20 0.41
MET P08581 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30194063 1.00 EPAS1 (0.44) EPAS1MAPK14MAP4K4TRPA1HSPB1
SCHEMBL21634034 0.88 EPAS1 (0.47) EPAS1MAPK14MAP4K4TRPA1HSPB1
SCHEMBL30194013 0.81 EPAS1 (0.41) EPAS1MAPK14MAP4K4TRPA1HSPB1
SCHEMBL30194117 0.78 AR (0.44) EPAS1TRPA1HSPB1
SCHEMBL28508478 0.78 GCK (0.47) EPAS1MAPK14TRPA1HSPB1
SCHEMBL28520346 0.78 AR (0.44) EPAS1TRPA1HSPB1
SCHEMBL16738742 0.78 EPAS1 (0.51) EPAS1MAPK14MAP4K4TRPA1HSPB1
SCHEMBL30194335 0.78 EPAS1 (0.51) EPAS1MAPK14MAP4K4TRPA1HSPB1
SCHEMBL190759 0.77 GCK (0.54) EPAS1
SCHEMBL16047284 0.76 EPAS1 (0.50) EPAS1MAPK14MAP4K4TRPA1HSPB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112300154-B Nitrogen-containing heterocyclic compound, preparation method and application thereof 上海弘翊生物科技有限公司 2023-01-24 CN disclosed
CN-112300154-A Nitrogen-containing heterocyclic compound, preparation method and application thereof 上海弘翊生物科技有限公司 2021-02-02 CN disclosed