SCHEMBL28515652

SCHEMBL28515652

C/C(=N/O)c1cc(C(=O)O)cc(Br)c1O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 2/20 0.58
AKR1C4 P17516 2/20 0.44
AKR1C3 P42330 2/20 0.44
AKR1C2 P52895 2/20 0.44
AKR1C1 Q04828 2/20 0.44
TPMT P51580 1/20 0.42
PTPN1 P18031 3/20 0.41
THRA P10827 1/20 0.39
THRB P10828 1/20 0.39
CA1 P00915 4/20 0.38
CA2 P00918 4/20 0.38
CA9 Q16790 4/20 0.38
CA4 P22748 3/20 0.38
CA12 O43570 3/20 0.38
CA7 P43166 3/20 0.38
CA14 Q9ULX7 3/20 0.38
CA3 P07451 2/20 0.38
CA6 P23280 2/20 0.38
CA5A P35218 2/20 0.38
CA5B Q9Y2D0 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21438414 1.00 TTR (0.58) TTRAKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL21545149 1.00 TTR (0.58) TTRAKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL29634023 0.83 KDM4E (0.46) TTRTPMTPTPN1CA1CA2
SCHEMBL21455367 0.83 KDM4E (0.46) TTRTPMTPTPN1CA1CA2
SCHEMBL28510333 0.83 KDM4E (0.46) TTRTPMTPTPN1CA1CA2
SCHEMBL1638962 0.82 TTR (0.67) TTRAKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL2439359 0.78 CA1 (0.46) TTRTPMTCA1CA2CA9
SCHEMBL2439356 0.78 CA1 (0.46) TTRTPMTCA1CA2CA9
SCHEMBL20870949 0.77 AKR1C4 (0.52) AKR1C4AKR1C3AKR1C2AKR1C1SMN1; SMN2
SCHEMBL1114408 0.75 TTR (1.00) TTRAKR1C4AKR1C3AKR1C2AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117164499-A Substituted benzofurans, benzopyrroles, benzothiophenes and structurally related complement inhibitors 拜奥克里斯特制药公司 2023-12-05 CN disclosed
CN-112272553-B Substituted benzofurans, benzopyrroles, benzothiophenes and structurally related complement inhibitors 拜奥克里斯特制药公司 2023-09-22 CN disclosed
CN-112272553-A Substituted benzofurans, benzopyrrole, benzothiophenes and structurally related complement inhibitors 拜奥克里斯特制药公司 2021-01-26 CN disclosed