SCHEMBL2851607

SCHEMBL2851607

CCCCc1ccc(C#Cc2ccc(CN(c3ccc(O)c(C(=O)O)c3)C(O)CCC3CCCC3)c(F)c2)cc1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.52
PTPRO Q16827 1/20 0.52
STAT3 P40763 8/20 0.39
KAT8 Q9H7Z6 2/20 0.36
UBLCP1 Q8WVY7 1/20 0.34
FFAR1 O14842 2/20 0.33
FFAR4 Q5NUL3 2/20 0.33
RARB P10826 2/20 0.32
BCHE P06276 1/20 0.32
ACHE P22303 1/20 0.32
RARA P10276 1/20 0.32
RARG P13631 1/20 0.32
MCL1 Q07820 1/20 0.32
HNF4A P41235 1/20 0.32
MEN1 O00255 1/20 0.31
RECQL P46063 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2853076 0.85 PTPN11 (0.53) PTPN11PTPROSTAT3KAT8MCL1
SCHEMBL2848964 0.76 PTPN11 (0.60) PTPN11PTPROSTAT3KAT8MCL1
SCHEMBL13711654 0.75 STAT3 (0.49) PTPN11PTPROSTAT3RARBRARA
SCHEMBL1736062 0.74 PTPN11 (0.55) PTPN11PTPROSTAT3KAT8MCL1
SCHEMBL1734720 0.73 PTPN11 (0.50) PTPN11PTPROSTAT3
SCHEMBL1733825 0.73 PTPN11 (0.58) PTPN11PTPROSTAT3RARBRARA
SCHEMBL1815749 0.72 PTPN11 (0.66) PTPN11PTPROSTAT3MCL1
SCHEMBL1734576 0.72 PTPN11 (0.62) PTPN11PTPROSTAT3KAT8MCL1
SCHEMBL1734722 0.72 PTPN11 (0.49) PTPN11PTPROSTAT3RARBRARA
SCHEMBL2853564 0.71 PTPN11 (0.51) PTPN11PTPROSTAT3KAT8FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654247-B1 ALKYNYL ARYL CARBOXAMIDES MERCK SERONO SA (CH) 2010-01-20 EP disclosed