SCHEMBL28516381

SCHEMBL28516381

CC1(Cn2cncn2)OC1c1ccc(Oc2ccccc2Cl)cc1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 6/20 0.41
KDM4E B2RXH2 4/20 0.36
CYP3A4 P08684 5/20 0.35
THRB P10828 1/20 0.35
DRD2 P14416 2/20 0.34
ALDH1A1 P00352 2/20 0.33
TSHR P16473 2/20 0.33
CYP2C9 P11712 1/20 0.33
ALOX15 P16050 1/20 0.32
NR1I2 O75469 1/20 0.32
LMNA P02545 1/20 0.32
FYN P06241 1/20 0.32
PGR P06401 1/20 0.32
HSP90AA1 P07900 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
CHRM5 P08912 1/20 0.32
ADRA2A P08913 1/20 0.32
CHRM1 P11229 1/20 0.32
ADRA2B P18089 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1280264 0.79 AR (0.42) ARKDM4ECYP3A4THRBALDH1A1
SCHEMBL16028244 0.71 CYP3A4 (0.58) KDM4ECYP3A4THRBALDH1A1TSHR
SCHEMBL28518928 0.71 AR (0.41) ARKDM4ECYP3A4ALDH1A1CYP2C9
SCHEMBL28516384 0.71 AR (0.43) ARKDM4ECYP3A4ALDH1A1TSHR
SCHEMBL1280154 0.71 CYP3A4 (0.55) KDM4ECYP3A4THRBTSHRCYP2C9
SCHEMBL1279694 0.70 CYP3A4 (0.52) KDM4ECYP3A4THRBTSHRCYP2C9
SCHEMBL1279615 0.70 CYP3A4 (0.47) KDM4ECYP3A4THRBTSHRCYP2C9
SCHEMBL28039664 0.67 KDM4E (0.43) ARKDM4EDRD2ALDH1A1TSHR
SCHEMBL1279614 0.67 CYP3A4 (0.53) ARKDM4ECYP3A4THRBTSHR
SCHEMBL22160949 0.67 MEN1 (0.39) CYP3A4THRBALDH1A1CYP2C9LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112047895-B Triazole compound, and preparation method and application thereof 东莞市东阳光农药研发有限公司 2024-05-14 CN disclosed
CN-112047895-A Triazole compound and preparation method and application thereof 东莞市东阳光农药研发有限公司 2020-12-08 CN disclosed