SCHEMBL28517569

SCHEMBL28517569

CCn1c(=O)c2[nH]c(C=Cc3cnc(OC)nc3)nc2n(CC)c1=O

nearest known ligand 0.70

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 1/20 0.47
SIRT1 Q96EB6 1/20 0.47
SIRT3 Q9NTG7 1/20 0.47
SIRT5 Q9NXA8 1/20 0.47
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
HPGD P15428 1/20 0.46
TSHR P16473 1/20 0.46
MAPK1 P28482 1/20 0.46
ADORA2B P29275 1/20 0.46
ADORA1 P30542 1/20 0.46
THPO P40225 1/20 0.46
PMP22 Q01453 1/20 0.46
HSD17B10 Q99714 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28517567 1.00 SIRT2 (0.47) SIRT2SIRT1SIRT3SIRT5KDM4E
SCHEMBL28528569 0.86 KDM4E (0.46) SIRT2SIRT1SIRT3SIRT5KDM4E
SCHEMBL30035898 0.86 KDM4E (0.46) SIRT2SIRT1SIRT3SIRT5KDM4E
SCHEMBL28528568 0.86 KDM4E (0.46) SIRT2SIRT1SIRT3SIRT5KDM4E
SCHEMBL7309870 0.84
SCHEMBL7309857 0.84
SCHEMBL7310644 0.81 ADORA2A (0.62) ADORA2BADORA1
SCHEMBL30632570 0.81 ADORA2A (0.62) ADORA2BADORA1
SCHEMBL7310635 0.81 ADORA2A (0.62) ADORA2BADORA1
SCHEMBL7311841 0.81 KDM4E (0.47) KDM4EALDH1A1CYP1A2CYP3A4HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112409360-A Heteroaryl vinyl xanthine derivatives and uses thereof 广东东阳光药业有限公司 2021-02-26 CN disclosed