SCHEMBL28524554

SCHEMBL28524554

CC(C)c1onc(-c2c(Cl)cccc2Cl)c1COc1ccc(COc2ccc(C(=O)O)cc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 20/20 1.00
LIFR P42702 3/20 1.00
PPARD Q03181 2/20 0.82

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30080745 0.97 NR1H4 (0.94) NR1H4LIFRPPARD
SCHEMBL30080655 0.97 NR1H4 (0.94) NR1H4LIFRPPARD
SCHEMBL21624446 0.96 NR1H4 (1.00) NR1H4LIFRPPARD
SCHEMBL10072267 0.93 NR1H4 (0.94) NR1H4LIFRPPARD
SCHEMBL30080609 0.92 NR1H4 (1.00) NR1H4LIFRPPARD
SCHEMBL30080781 0.92 NR1H4 (0.86) NR1H4LIFRPPARD
SCHEMBL28908463 0.92 NR1H4 (0.86) NR1H4LIFRPPARD
SCHEMBL14279685 0.90 NR1H4 (0.82) NR1H4LIFRPPARD
SCHEMBL28529145 0.90 NR1H4 (1.00) NR1H4LIFRPPARD
SCHEMBL30080791 0.90 NR1H4 (0.95) NR1H4LIFRPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3823960-B1 ISOXAZOLE AS FXR RECEPTOR AGONISTS BAR PHARMACEUTICALS SOC A RESPONSABILITA LIMITATA (IT) 2022-09-14 EP disclosed
CN-112424173-A Isoxazoles as FXR receptor agonists 巴尔制药有限公司 2021-02-26 CN disclosed