SCHEMBL28527217

SCHEMBL28527217

NNC(=O)C1CCC(OC(N)=O)CC1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.36
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
KMT2A Q03164 1/20 0.31
POLB P06746 1/20 0.31
HDAC8 Q9BY41 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
MAPK10 P53779 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28527216 1.00 ATM (0.36) ATMLMNAMAPTSMN1; SMN2NPSR1
SCHEMBL16335867 0.81 ATM (0.38) ATMSMN1; SMN2KMT2APOLBMAPK10
SCHEMBL21378960 0.81 POLB (0.48) ATMLMNAPOLB
SCHEMBL16335866 0.81 ATM (0.38) ATMSMN1; SMN2KMT2APOLBMAPK10
SCHEMBL425737 0.80
SCHEMBL29222629 0.80 HDAC8 (0.42) LMNAMAPTKMT2APOLBHDAC8
SCHEMBL363166 0.80
SCHEMBL1142180 0.80 HDAC8 (0.42) LMNAMAPTKMT2APOLBHDAC8
SCHEMBL15656336 0.79 GAA (0.41) ATMMAPTSMN1; SMN2KMT2APOLB
SCHEMBL29148774 0.79 GAA (0.41) ATMMAPTSMN1; SMN2KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112566915-A Thiadiazole IRAK4 inhibitor 吉利德科学公司 2021-03-26 CN disclosed
CN-112566697-A Pyrrolo [1,2-b ] pyridazine derivatives as IRAK4 inhibitors 吉利德科学公司 2021-03-26 CN disclosed
CN-112533924-A Pyrrolo [1,2-b ] pyridazine derivatives as IRAK4 inhibitors 吉利德科学公司 2021-03-19 CN disclosed