SCHEMBL28527474

SCHEMBL28527474

COC(=O)NC1CC(NC(=O)OC(C)(C)C)C1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.56
CTSK P43235 2/20 0.47
GAA P10253 2/20 0.46
KMT2A Q03164 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
NFKB1 P19838 1/20 0.45
NFKB2 Q00653 1/20 0.45
RELA Q04206 1/20 0.45
KDM1A O60341 2/20 0.44
MAOB P27338 1/20 0.44
EPHX2 P34913 1/20 0.44
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CYP2C9 P11712 1/20 0.43
HSD11B1 P28845 1/20 0.43
EPHX1 P07099 1/20 0.41
MEN1 O00255 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31246211 0.87 BTK (0.51) BTKCTSKGAAKMT2AL3MBTL1
SCHEMBL18696405 0.86 BTK (0.54) BTKCTSKGAAKMT2AL3MBTL1
SCHEMBL31246148 0.86 BTK (0.54) BTKCTSKGAAKMT2AL3MBTL1
SCHEMBL18617791 0.86 BTK (0.54) BTKCTSKGAAKMT2AL3MBTL1
SCHEMBL16748085 0.86 BTK (0.54) BTKCTSKGAAKMT2AL3MBTL1
SCHEMBL26985685 0.86 BTK (0.54) BTKCTSKGAAKMT2AL3MBTL1
SCHEMBL31246132 0.86 BTK (0.54) BTKCTSKGAAKMT2AL3MBTL1
SCHEMBL11901905 0.85 BTK (0.53) BTKCTSKGAAKMT2AL3MBTL1
SCHEMBL11901221 0.85 BTK (0.53) BTKCTSKGAAKMT2AL3MBTL1
SCHEMBL11901219 0.85 BTK (0.53) BTKCTSKGAAKMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106188027-B Aromatic heterocyclic derivative and application thereof in medicine 广东东阳光药业有限公司 2020-10-20 CN disclosed