SCHEMBL28528554

SCHEMBL28528554

COCCOc1ccc([N+](=O)[O-])c(C(=O)O)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.49
DTYMK P23919 1/20 0.49
KMT2A Q03164 4/20 0.48
MEN1 O00255 3/20 0.48
HTT P42858 1/20 0.48
MAPT P10636 4/20 0.48
ALDH1A1 P00352 6/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
AKR1C3 P42330 3/20 0.46
AKR1C2 P52895 3/20 0.46
AKR1C1 Q04828 2/20 0.46
AKR1B10 O60218 1/20 0.46
AKR1B1 P15121 1/20 0.46
AKR1C4 P17516 1/20 0.46
TTR P02766 1/20 0.46
PPOX P50336 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
HCAR3 P49019 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30686065 1.00 KDM4E (0.49) KDM4EDTYMKKMT2AMEN1HTT
SCHEMBL3512088 0.89 AKR1C3 (0.46) KDM4EKMT2AMEN1HTTMAPT
SCHEMBL30686032 0.88 MAPT (0.47) KDM4EKMT2AMEN1HTTMAPT
SCHEMBL28528923 0.88 MAPT (0.47) KDM4EKMT2AMEN1HTTMAPT
SCHEMBL268658 0.88 TDP1 (0.55) KDM4EKMT2AMEN1HTTMAPT
SCHEMBL26343197 0.87 DTYMK (0.50) KDM4EDTYMKKMT2AMEN1HTT
SCHEMBL2155062 0.87 MAPT (0.63) KDM4EDTYMKKMT2AMEN1HTT
SCHEMBL8381314 0.87 MAPT (0.56) KDM4EDTYMKKMT2AMEN1HTT
SCHEMBL21707908 0.86 TSHR (0.48) KDM4EKMT2AMEN1HTTMAPT
SCHEMBL8872227 0.84 MAPT (0.61) KDM4EDTYMKKMT2AMEN1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112409332-B Triazole derivative and application thereof in medicines 广东东阳光药业股份有限公司 2023-12-08 CN disclosed
CN-112409332-A Triazole derivative and application thereof in medicines 广东东阳光药业有限公司 2021-02-26 CN disclosed