SCHEMBL28529932

SCHEMBL28529932

CC(C)(C)OC(=O)NC1CCC(Oc2cc(F)c(F)c(F)c2)C1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.44
KDM1A O60341 1/20 0.42
MAOB P27338 1/20 0.42
PIK3CD O00329 1/20 0.40
ACACB O00763 2/20 0.40
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
PARP1 P09874 1/20 0.39
GPR119 Q8TDV5 1/20 0.39
EPHX2 P34913 2/20 0.38
KMT2A Q03164 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KAT6A Q92794 1/20 0.38
KAT5 Q92993 1/20 0.38
DRD2 P14416 2/20 0.38
JAK2 O60674 3/20 0.37
JAK1 P23458 3/20 0.37
CTSK P43235 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21503612 1.00 BTK (0.44) BTKKDM1AMAOBPIK3CDACACB
SCHEMBL28529931 1.00 BTK (0.44) BTKKDM1AMAOBPIK3CDACACB
SCHEMBL24975362 0.91 BTK (0.41) BTKKDM1AMAOBPIK3CDNFKB1
SCHEMBL29279741 0.91 BTK (0.41) BTKKDM1AMAOBPIK3CDNFKB1
SCHEMBL29874615 0.84 PIK3CD (0.39) BTKKDM1AMAOBPIK3CDNFKB1
SCHEMBL29874623 0.82 PIK3CD (0.41) BTKKDM1AMAOBPIK3CDNFKB1
SCHEMBL21492528 0.82 EPHX2 (0.43) EPHX2
SCHEMBL21492525 0.82 EPHX2 (0.43) EPHX2
SCHEMBL29874307 0.81 BTK (0.39) BTKKDM1AMAOBPIK3CDNFKB1
SCHEMBL29874542 0.81 FFAR4 (0.39) BTKKDM1AMAOBPIK3CDNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112218865-A Pteridinone compounds and uses thereof 沃泰克斯药物股份有限公司 2021-01-12 CN disclosed