SCHEMBL28533709

SCHEMBL28533709

CC(C)(C)OC(=O)C=C1CCn2c1cc1cc(O)ccc12

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.39
CLK1 P49759 1/20 0.33
DYRK1A Q13627 1/20 0.33
DYRK1B Q9Y463 1/20 0.33
NR1H2 P55055 1/20 0.33
HTR6 P50406 1/20 0.32
GAA P10253 2/20 0.31
MAPK1 P28482 1/20 0.31
ALOX5 P09917 1/20 0.30
ALDH1A1 P00352 1/20 0.30
ALOX15 P16050 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14327924 0.88 NR1H2 (0.36) NR1H2ALOX5MEN1KMT2A
SCHEMBL2013305 0.87 MCL1 (0.38) NR1H2
SCHEMBL2013306 0.87 MCL1 (0.38) NR1H2
SCHEMBL2447541 0.82 SRD5A2 (0.49) ALOX5ALDH1A1MEN1KMT2A
SCHEMBL2447542 0.82 SRD5A2 (0.49) ALOX5ALDH1A1MEN1KMT2A
SCHEMBL2021474 0.82 SRD5A2 (0.49) ALOX5ALDH1A1MEN1KMT2A
SCHEMBL2014413 0.81 CLK1 (0.32) CLK1DYRK1ADYRK1BGAAMAPK1
SCHEMBL2014416 0.81 CLK1 (0.32) CLK1DYRK1ADYRK1BGAAMAPK1
SCHEMBL2017568 0.80 PRMT5 (0.37)
SCHEMBL2017566 0.80 PRMT5 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105816453-B Substituted tricyclic acid derivatives as S1P1 receptor agonists for the treatment of autoimmune and inflammatory disorders 艾尼纳制药公司 2021-03-05 CN disclosed