SCHEMBL28543731

SCHEMBL28543731

O=C(O)c1cnn2ccc(O)cc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHB3 P54753 7/20 0.41
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA7 P43166 2/20 0.40
CA9 Q16790 2/20 0.40
CA14 Q9ULX7 2/20 0.40
ALDH1A1 P00352 2/20 0.40
ALOX5 P09917 1/20 0.40
PTGS2 P35354 1/20 0.40
TSHR P16473 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CAMKK1 Q8N5S9 2/20 0.38
CAMKK2 Q96RR4 2/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TGFBR1 P36897 2/20 0.37
KDM4E B2RXH2 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3606337 0.85 NPC1 (0.45) EPHB3ALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL13954506 0.81 MAPT (0.41) EPHB3ALDH1A1PTGS2L3MBTL1CAMKK1
SCHEMBL12477928 0.81 EPHB3 (0.43) EPHB3L3MBTL1CAMKK1CAMKK2TGFBR1
SCHEMBL3073610 0.81 EPHB3 (0.56) EPHB3ALDH1A1L3MBTL1TGFBR1KDM4E
SCHEMBL31547078 0.81 IRAK4 (0.41) EPHB3ALDH1A1L3MBTL1CAMKK1CAMKK2
SCHEMBL24369482 0.81 EPHB3 (0.59) EPHB3CA1CA2ALDH1A1TSHR
SCHEMBL3089211 0.81 EIF4A3 (0.45) EPHB3L3MBTL1CAMKK1CAMKK2NPC1
SCHEMBL3612196 0.81 CA12 (0.46) EPHB3CA12CA1CA2CA7
SCHEMBL29014099 0.79 NPC1 (0.49) EPHB3ALDH1A1L3MBTL1NPC1RAB9A
SCHEMBL23872949 0.78 TDP1 (0.40) EPHB3L3MBTL1CAMKK1CAMKK2TGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108699038-B Spirocyclic heptane salicylamides and related compounds as Rock inhibitors 百时美施贵宝公司 2021-04-16 CN disclosed