SCHEMBL28544019

SCHEMBL28544019

CN(C(=O)Oc1cc(NC(=O)c2c[nH]c3ccccc3c2=O)ccc1C(C)(C)C)C(C)(C)C

nearest known ligand 0.69

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CFTR P13569 19/20 0.69
ADORA3 P0DMS8 1/20 0.56
ADRB3 P13945 1/20 0.56
TBXA2R P21731 1/20 0.56
SLC6A2 P23975 1/20 0.56
AGTR1 P30556 1/20 0.56
MC4R P32245 1/20 0.56
PTGS2 P35354 1/20 0.56
SLC6A3 Q01959 1/20 0.56
MAOB P27338 1/20 0.55
GABRA1 P14867 1/20 0.53
GABRB1 P18505 1/20 0.53
GABRA5 P31644 1/20 0.53
GABRA3 P34903 1/20 0.53
GABRA2 P47869 1/20 0.53
GABRB2 P47870 1/20 0.53
GABRA4 P48169 1/20 0.53
GABRA6 Q16445 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL396856 0.87 CFTR (0.76) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL396475 0.83 CFTR (0.76) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL399248 0.83 CFTR (0.72) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL396079 0.82 CFTR (1.00) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL395729 0.82 CFTR (1.00) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL396505 0.81 CFTR (0.67) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL397109 0.81 CFTR (0.76) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL2976145 0.81 CFTR (1.00) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL397527 0.81 CFTR (1.00) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL395014 0.81 CFTR (0.66) CFTRADORA3ADRB3TBXA2RSLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107501099-B Modulators of ATP-binding cassette transporters 沃泰克斯药物股份有限公司 2021-03-19 CN disclosed