SCHEMBL28544845

SCHEMBL28544845

COc1ccnc(NC2CCCN(C(=O)OC(C)(C)C)C2)n1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CDK12 Q9NYV4 3/20 0.60
CCNK O75909 2/20 0.49
USP30 Q70CQ3 3/20 0.48
PIK3CD O00329 1/20 0.47
BTK Q06187 3/20 0.47
TRPV1 Q8NER1 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
PARP1 P09874 1/20 0.45
ALDH1A1 P00352 1/20 0.44
ANO1 Q5XXA6 1/20 0.43
GPR119 Q8TDV5 1/20 0.43
PIM1 P11309 2/20 0.42
PIM2 Q9P1W9 2/20 0.42
EGFR P00533 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23292284 1.00 CDK12 (0.60) CDK12CCNKUSP30PIK3CDBTK
SCHEMBL22895718 1.00 CDK12 (0.60) CDK12CCNKUSP30PIK3CDBTK
SCHEMBL28550665 0.89 CDK12 (0.60) CDK12CCNKUSP30BTKTRPV1
SCHEMBL23292355 0.89 CDK12 (0.60) CDK12CCNKUSP30BTKTRPV1
SCHEMBL22895525 0.89 CDK12 (0.60) CDK12CCNKUSP30BTKTRPV1
SCHEMBL22895338 0.84 CDK12 (0.59) CDK12CCNKUSP30PIK3CDBTK
SCHEMBL23292383 0.84 CDK12 (0.59) CDK12CCNKUSP30PIK3CDBTK
SCHEMBL9942554 0.84 USP30 (0.46) CDK12USP30PIK3CDBTKTRPV1
SCHEMBL9899889 0.84 USP30 (0.46) CDK12USP30PIK3CDBTKTRPV1
SCHEMBL28571259 0.82 BTK (0.43) CDK12CCNKUSP30PIK3CDBTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112638373-A Cyclin-dependent kinase inhibitors 金耐特生物制药公司 2021-04-09 CN disclosed