SCHEMBL28546348

SCHEMBL28546348

Cc1cnc(Nc2cc(CN3CCOCC3)cc(N[C@H]3CCCN(C(=O)O)C3)n2)s1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 1/20 0.46
BTK Q06187 5/20 0.45
HCK P08631 3/20 0.45
ITK Q08881 2/20 0.42
KDR P35968 5/20 0.40
LCK P06239 1/20 0.39
AURKB Q96GD4 1/20 0.39
CNR2 P34972 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CHEK1 O14757 1/20 0.37
JAK3 P52333 1/20 0.37
JAK2 O60674 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28554401 1.00 MAP3K12 (0.46) MAP3K12BTKHCKITKKDR
SCHEMBL21777160 0.91 BTK (0.54) MAP3K12BTKHCKITKJAK3
SCHEMBL21777159 0.91 BTK (0.54) MAP3K12BTKHCKITKJAK3
SCHEMBL23608029 0.91 BTK (0.54) MAP3K12BTKHCKITKJAK3
SCHEMBL30167089 0.91 BTK (0.54) MAP3K12BTKHCKITKJAK3
Hydrochloric Acid SCHEMBL23608055 0.91 BTK (0.54) MAP3K12BTKHCKITKJAK3
Hydrochloric Acid SCHEMBL23607999 0.91 BTK (0.54) MAP3K12BTKHCKITKJAK3
SCHEMBL23608042 0.90 BTK (0.44) MAP3K12BTKHCKITKKDR
SCHEMBL23608053 0.90 BTK (0.47) MAP3K12BTKHCKITKKDR
SCHEMBL23608033 0.90 BTK (0.43) MAP3K12BTKHCKITKKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112638910-B New heterocyclic amine derivatives and pharmaceutical compositions containing the same 株式会社大熊制药 2024-06-11 CN disclosed
CN-112638910-A Novel heterocyclic amine derivatives and pharmaceutical compositions comprising the same 株式会社大熊制药 2021-04-09 CN disclosed