SCHEMBL28558647

SCHEMBL28558647

Cc1cc2cccc(C#N)c2cn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.49
CYP1A2 P05177 1/20 0.48
CYP2A6 P11509 1/20 0.48
TGFBR1 P36897 1/20 0.41
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
HPGDS O60760 1/20 0.39
GABRA1 P14867 2/20 0.39
GABRG2 P18507 2/20 0.39
GABRB3 P28472 2/20 0.39
GABRA2 P47869 2/20 0.39
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
TSHR P16473 1/20 0.38
NCOA3 Q9Y6Q9 1/20 0.38
GRM5 P41594 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2749751 0.79 HTT (0.49) HTTTGFBR1CA1CA2MAPT
SCHEMBL8404524 0.76 CYP1A2 (0.57) CYP1A2CYP2A6MAPTTDP1TSHR
SCHEMBL29404615 0.76 CYP1A2 (0.57) CYP1A2CYP2A6MAPTTDP1TSHR
SCHEMBL18322219 0.75 HTT (0.53) HTTCA1CA2MAPTTSHR
Ammonia Solution, Strong SCHEMBL28514949 0.74 CYP1A2 (0.55) CYP1A2CYP2A6MAPTTDP1TSHR
SCHEMBL818940 0.73 HTT (0.52) HTTCYP1A2CA1CA2MAPT
SCHEMBL9226415 0.73 CYP1A2 (0.57) HTTCYP1A2CYP2A6CA1CA2
SCHEMBL28474208 0.73 CYP1A2 (0.53) HTTCYP1A2CYP2A6MAPTKDM4E
SCHEMBL16168207 0.73 CYP1A2 (0.53) CYP1A2CYP2A6MAPTKMT2ANPSR1
SCHEMBL1564051 0.73 IDO1 (0.57) CYP1A2CYP2A6MEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112121463-B Preparation method of polysubstituted benzo nitrogen-containing heterocyclic methylamine 烟台宁远药业有限公司 2022-03-22 CN claimed
CN-112121463-A Preparation method of polysubstituted benzo nitrogen-containing heterocyclic methylamine 烟台宁远药业有限公司 2020-12-25 CN claimed
CN-112121463-B Preparation method of polysubstituted benzo nitrogen-containing heterocyclic methylamine 烟台宁远药业有限公司 2022-03-22 CN disclosed
CN-112121463-A Preparation method of polysubstituted benzo nitrogen-containing heterocyclic methylamine 烟台宁远药业有限公司 2020-12-25 CN disclosed