SCHEMBL28565745

SCHEMBL28565745

NC(=O)c1cc(-c2cc(Cl)cc(Cl)c2)ccc1NC1CCC(O)CC1

nearest known ligand 0.71

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 4/20 0.71
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA3 P07451 1/20 0.41
CA6 P23280 1/20 0.41
CA7 P43166 1/20 0.41
CA5B Q9Y2D0 1/20 0.41
TP53 P04637 1/20 0.41
MDM2 Q00987 1/20 0.41
ROCK2 O75116 1/20 0.40
BMPR1B O00238 1/20 0.40
BMPR1A P36894 1/20 0.40
TGFBR1 P36897 1/20 0.40
ACVRL1 P37023 1/20 0.40
ACVR1 Q04771 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28565744 1.00 HSP90AA1 (0.71) HSP90AA1CA1CA2CA3CA6
SCHEMBL28568960 0.88 HSP90AA1 (0.74) HSP90AA1CA1CA2CA3CA6
SCHEMBL28568961 0.88 HSP90AA1 (0.74) HSP90AA1CA1CA2CA3CA6
SCHEMBL28562475 0.85 HSP90AA1 (0.65) HSP90AA1CA1CA2CA3CA6
SCHEMBL28562473 0.85 HSP90AA1 (0.65) HSP90AA1CA1CA2CA3CA6
SCHEMBL28568011 0.85 HSP90AA1 (0.71) HSP90AA1
SCHEMBL28568013 0.85 HSP90AA1 (0.71) HSP90AA1
SCHEMBL28565743 0.85 HSP90AA1 (0.74) HSP90AA1
SCHEMBL28565741 0.85 HSP90AA1 (0.74) HSP90AA1
SCHEMBL28572877 0.82 HSP90AA1 (0.71) HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108147978-B Grp94 inhibitor with benzamide parent nucleus structure and application thereof 中国药科大学 2021-05-07 CN disclosed