SCHEMBL28565798

SCHEMBL28565798

O=C(O)CC[C@H](c1cccc(Cl)c1)[C@@H](O)c1ccc(Cl)cn1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 7/20 0.45
S1PR4 O95977 5/20 0.45
S1PR2 O95136 4/20 0.45
ADRB2 P07550 3/20 0.40
ADRB1 P08588 3/20 0.40
ADRB3 P13945 3/20 0.40
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
FOLH1 Q04609 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9993528 1.00 S1PR3 (0.45) S1PR3S1PR4S1PR2ADRB2ADRB1
SCHEMBL28565309 1.00 S1PR3 (0.45) S1PR3S1PR4S1PR2ADRB2ADRB1
SCHEMBL9993134 0.86 S1PR3 (0.44) S1PR3S1PR4S1PR2ADRB2ADRB1
SCHEMBL9990779 0.86 S1PR3 (0.44) S1PR3S1PR4S1PR2ADRB2ADRB1
SCHEMBL9990780 0.86 S1PR3 (0.44) S1PR3S1PR4S1PR2ADRB2ADRB1
SCHEMBL24714159 0.82 SLC6A2 (0.47) ADRB2ADRB1ADRB3MEN1KMT2A
SCHEMBL28578802 0.82 SLC6A2 (0.47) ADRB2ADRB1ADRB3MEN1KMT2A
SCHEMBL9992346 0.82 SLC6A2 (0.47) ADRB2ADRB1ADRB3MEN1KMT2A
SCHEMBL28574464 0.81 S1PR3 (0.40) S1PR3S1PR4S1PR2ADRB2ADRB1
SCHEMBL28571545 0.81 S1PR3 (0.40) S1PR3S1PR4S1PR2ADRB2ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105153014-B Piperidinone derivatives as MDM2 inhibitors for the treatment of cancer 安姆根有限公司 2021-06-01 CN disclosed