SCHEMBL28566581

SCHEMBL28566581

O=[N+]([O-])c1c(CCc2ccccc2)ccc2ccccc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.53
CYP3A4 P08684 1/20 0.50
ALDH1A1 P00352 3/20 0.42
MAPT P10636 4/20 0.42
HPGD P15428 3/20 0.42
HTT P42858 2/20 0.42
NPC1 O15118 1/20 0.42
LMNA P02545 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
NCEH1 Q6PIU2 1/20 0.42
HPRT1 P00492 1/20 0.41
HSP90AA1 P07900 2/20 0.40
CRHBP P24387 1/20 0.40
CRHR2 Q13324 1/20 0.40
GAA P10253 2/20 0.40
PIN1 Q13526 1/20 0.40
CYP1A1 P04798 1/20 0.39
CYP1B1 Q16678 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8576110 0.83 TSHR (0.58) TSHRCYP3A4ALDH1A1MAPTNCEH1
SCHEMBL7057106 0.83 TSHR (0.54) TSHRCYP3A4ALDH1A1MAPTNCEH1
SCHEMBL9638921 0.81 TSHR (0.53) TSHRCYP3A4ALDH1A1MAPTNCEH1
SCHEMBL12363753 0.80 TSHR (0.64) TSHRCYP3A4ALDH1A1MAPTHPGD
SCHEMBL2888432 0.80 TSHR (0.59) TSHRCYP3A4ALDH1A1MAPTNCEH1
SCHEMBL29844402 0.79 TSHR (0.57) TSHRCYP3A4ALDH1A1MAPTHTT
SCHEMBL11350432 0.79 TSHR (0.57) TSHRCYP3A4ALDH1A1MAPTHTT
SCHEMBL7061346 0.78 MAPT (0.41) TSHRCYP3A4ALDH1A1MAPTHPGD
SCHEMBL31146864 0.78 TSHR (0.53) TSHRCYP3A4ALDH1A1MAPTHPGD
SCHEMBL28965419 0.78 TSHR (0.53) TSHRCYP3A4ALDH1A1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112047871-B Preparation method of indole compound 南京大学 2022-06-21 CN disclosed
CN-112047871-A Preparation method of indole compound 南京大学 2020-12-08 CN disclosed