SCHEMBL2856982

SCHEMBL2856982

Cc1cc(CC(C(=O)O)C(=O)O)cc(C(C)(C)C)c1O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.49
CYP2C9 P11712 2/20 0.49
CYP2C19 P33261 2/20 0.49
HMGCR P04035 2/20 0.44
GLRA3 O75311 1/20 0.43
GLRB P48167 1/20 0.43
KMT2A Q03164 6/20 0.41
MEN1 O00255 5/20 0.41
ALDH1A1 P00352 4/20 0.41
TSHR P16473 3/20 0.41
CYP3A4 P08684 2/20 0.41
MAPK1 P28482 2/20 0.41
BLM P54132 2/20 0.41
ATM Q13315 2/20 0.41
HIF1A Q16665 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
USP2 O75604 1/20 0.41
CYP2D6 P10635 1/20 0.41
MAPT P10636 1/20 0.41
GAA P10253 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2671331 0.90 HMGCR (0.53) CYP1A2CYP2C9CYP2C19HMGCRGLRA3
SCHEMBL10793871 0.89 CYP1A2 (0.47) CYP1A2CYP2C9CYP2C19HMGCRGLRA3
SCHEMBL8336608 0.88 CYP1A2 (0.46) CYP1A2CYP2C9CYP2C19HMGCRGLRA3
SCHEMBL29228065 0.86 CYP1A2 (0.45) CYP1A2CYP2C9CYP2C19HMGCRGLRA3
SCHEMBL11490153 0.86 CYP1A2 (0.45) CYP1A2CYP2C9CYP2C19HMGCRGLRA3
SCHEMBL11854423 0.85 HMGCR (0.44) CYP1A2CYP2C9CYP2C19HMGCRKMT2A
SCHEMBL6714136 0.84 CYP1A2 (0.42) CYP1A2CYP2C9CYP2C19HMGCRGLRA3
SCHEMBL2133313 0.83 CYP1A2 (0.41) CYP1A2CYP2C9CYP2C19HMGCRGLRA3
SCHEMBL5817828 0.82 CYP1A2 (0.41) CYP1A2CYP2C9CYP2C19HMGCRGLRA3
SCHEMBL7603596 0.81 ESR1 (0.47) HMGCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 484 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0335262-B1 Phosphite compounds YOSHITOMI PHARMACEUTICAL (JP) 1995-05-31 EP claimed
EP-0335262-A2 Phosphite compounds YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1989-10-04 EP claimed
US-4221701-A ESTERS OF TETRAMETHYLPIPERIDINOL WITH HYDROXYBENZYLMALONIC ACID CIBA-GEIGY CORPORATION (US) 1980-09-09 US claimed
US-3993655-A ESTERS OF TETRAMETHYLPIPERIDINOLS CIBA-GEIGY CORPORATION (US) 1976-11-23 US claimed
EP-3194482-B1 USE OF PHOSPHOROUS-CONTAINING ORGANIC OXYIMIDES AS FLAME RETARDANTS FOR PLASTICS, FLAME-RETARDANT PLASTIC COMPOSITIONS, METHOD FOR THE PRODUCTION THEREOF, MOULDED PART, PAINT AND COATINGS FRAUNHOFER GES FORSCHUNG (DE) 2024-05-08 EP disclosed
WO-2024062815-A1 AROMATIC POLYCARBONATE RESIN COMPOSITION AND MOLDED ARTICLE THEREOF 帝人株式会社 2024-03-28 WO disclosed
EP-3710424-B1 COMPOUNDS HAVING A STABILIZING EFFECT, METHOD FOR PRODUCING SAID COMPOUNDS, COMPOSITION CONTAINING SAID STABILIZING COMPOUNDS, METHOD FOR STABILIZING AN ORGANIC COMPONENT, AND USE OF STABILIZING COMPOUNDS FRAUNHOFER GES FORSCHUNG (DE) 2024-01-03 EP disclosed
EP-3947540-B1 METHOD FOR STABILIZING THERMOPLASTIC RECYCLATES, STABILIZED PLASTIC COMPOSITIONS, AND MOLDING COMPOUNDS AND MOLDED PARTS PRODUCED THEREFROM FRAUNHOFER GES FORSCHUNG (DE) 2023-08-16 EP disclosed
WO-2023120669-A1 CYCLOOLEFIN COPOLYMER, RESIN COMPOSITION, AND FILM- OR SHEET-SHAPED ARTICLE ポリプラスチックス株式会社 2023-06-29 WO disclosed
US-11347146-B2 Resin composition TORAY INDUSTRIES, INC. (JP) 2022-05-31 US disclosed
CN-111511558-A Multilayer body 帝人株式会社 2020-08-07 CN disclosed
CN-105693698-B Multi-functional hindered amine light stabilizer 巴斯夫欧洲公司 2019-11-22 CN disclosed
US-4405737-A OLEFIN STABILIZERS ADEKA ARGUS CHEMICAL CO., LTD. (JP) 1983-09-20 US disclosed
EP-0066621-A4 HINDERED PHENOLIC ANTIOXIDANTS AND DIAZACYCLOALKANE UV STABILIZERS IN POLYMERIC FILMS. GOODRICH CO B F (US) 1983-06-08 EP disclosed
US-4371651-A PHOTOSTABILITY, HEAT RESISTANCE PHOENIX CHEMICAL CORPORATION (US) 1983-02-01 US disclosed
EP-0066621-A1 HINDERED PHENOLIC ANTIOXIDANTS AND DIAZACYCLOALKANE UV STABILIZERS IN POLYMERIC FILMS. GOODRICH CO B F (US) 1982-12-15 EP disclosed
WO-1982002169-A1 HINDERED PHENOLIC ANTIOXIDANTS AND DIAZACYCLOALKANE UV STABILIZERS IN POLYMERIC FILMS KLETECKA GEORGE 1982-07-08 WO disclosed
US-4125516-A HEAT STABILIZER, ANTIOXIDANT, DISCOLORATION INHIBITON CIBA-GEIGY CORPORATION (US) 1978-11-14 US disclosed
US-4093586-A Pyrrolidine dicarboxylic acids and esters and stabilized compositions CIBA-GEIGY CORPORATION (US) 1978-06-06 US disclosed
US-3950382-A STABILIZERS FOR POLYOLEFINS CIBA-GEIGY CORPORATION (US) 1976-04-13 US disclosed