SCHEMBL28574656

SCHEMBL28574656

CC(=O)SCCCCCCNC(=O)c1n[nH]c2c1CCc1c-2cnn1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
HTR1A P08908 7/20 0.33
DRD2 P14416 6/20 0.33
HTR2A P28223 6/20 0.33
GSK3B P49841 1/20 0.31
DYRK1A Q13627 1/20 0.31
FOLH1 Q04609 1/20 0.31
CYP2D6 P10635 1/20 0.31
THRB P10828 3/20 0.30
LMNA P02545 2/20 0.30
HTR3E A5X5Y0 1/20 0.30
HTR3B O95264 1/20 0.30
HTR3A P46098 1/20 0.30
HTR3D Q70Z44 1/20 0.30
HTR3C Q8WXA8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28568974 0.89 HDAC3 (0.35) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL28576385 0.88 HDAC6 (0.35) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL28587599 0.87 HDAC6 (0.42) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL28582693 0.86 HDAC3 (0.33) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL28576387 0.86 HDAC3 (0.33) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL28576560 0.86 HDAC3 (0.34) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL28573732 0.85 ITK (0.36) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL28576561 0.85 HDAC3 (0.33) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL28587603 0.84 HDAC3 (0.34) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL28575703 0.84 CCNA2 (0.39) HDAC3HDAC4HDAC1HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109384793-B Thiol compound with HDAC6 inhibitory activity and application thereof 沈阳药科大学 2021-05-07 CN claimed
CN-109384793-B Thiol compound with HDAC6 inhibitory activity and application thereof 沈阳药科大学 2021-05-07 CN disclosed