SCHEMBL28577358

SCHEMBL28577358

COc1cc(NC(=O)c2ccnc3ccc(Cl)cc23)ccc1NC(=O)c1cccc(Cl)c1

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.59
MAPT P10636 2/20 0.59
POLB P06746 1/20 0.59
GRM5 P41594 1/20 0.54
GRM4 Q14833 5/20 0.52
KDR P35968 4/20 0.51
KMT2A Q03164 3/20 0.48
MEN1 O00255 2/20 0.48
RAB9A P51151 2/20 0.48
NPC1 O15118 1/20 0.48
TP53 P04637 1/20 0.48
ALDH1A1 P00352 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29886473 1.00 KDM4E (0.59) KDM4EMAPTPOLBGRM5GRM4
SCHEMBL28589498 0.93 KDM4E (0.56) KDM4EMAPTPOLBGRM5GRM4
SCHEMBL29886248 0.93 KDM4E (0.56) KDM4EMAPTPOLBGRM5GRM4
SCHEMBL29886583 0.93 KDM4E (0.56) KDM4EMAPTPOLBGRM5GRM4
SCHEMBL29886180 0.93 KDM4E (0.59) KDM4EMAPTPOLBGRM5GRM4
SCHEMBL28579647 0.93 KDM4E (0.59) KDM4EMAPTPOLBGRM5GRM4
SCHEMBL29886104 0.82 GRM5 (0.65) KDM4EMAPTPOLBGRM5GRM4
SCHEMBL28577355 0.82 GRM5 (0.65) KDM4EMAPTPOLBGRM5GRM4
SCHEMBL28587976 0.73 POLB (0.63) KDM4EMAPTPOLBGRM5KMT2A
SCHEMBL16431420 0.72 GRM5 (0.65) KDM4EMAPTPOLBGRM5KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113061098-B Amide compound and derivative thereof, preparation method, pharmaceutical composition and application 中国药科大学 2022-08-30 CN claimed
CN-113061098-A Amide compound and derivative thereof, preparation method, pharmaceutical composition and application 中国药科大学 2021-07-02 CN claimed
CN-113061098-B Amide compound and derivative thereof, preparation method, pharmaceutical composition and application 中国药科大学 2022-08-30 CN disclosed
CN-113061098-A Amide compound and derivative thereof, preparation method, pharmaceutical composition and application 中国药科大学 2021-07-02 CN disclosed