SCHEMBL28579641

SCHEMBL28579641

COCCn1cc2c(n1)CCc1c(C(=O)NCCCCCCSC(C)=O)n[nH]c1-2

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 4/20 0.41
HDAC6 Q9UBN7 2/20 0.37
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
LMNA P02545 1/20 0.37
THRB P10828 1/20 0.37
KDM4E B2RXH2 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
GAA P10253 1/20 0.32
HTR1A P08908 4/20 0.31
HTR2A P28223 4/20 0.31
DRD2 P14416 3/20 0.31
HTR2C P28335 2/20 0.31
HRH1 P35367 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28568420 0.93 HDAC3 (0.36) IKBKBHDAC6HDAC3HDAC4HDAC1
SCHEMBL28582772 0.90 HDAC3 (0.37) IKBKBHDAC6HDAC3HDAC4HDAC1
SCHEMBL28576372 0.89 HDAC3 (0.40) HDAC6HDAC3HDAC4HDAC1HDAC2
SCHEMBL28580756 0.88 HDAC3 (0.35) IKBKBHDAC6HDAC3HDAC4HDAC1
SCHEMBL28568413 0.88 IKBKB (0.43) IKBKBHDAC6HDAC3HDAC4HDAC1
SCHEMBL28583307 0.86 SMN1; SMN2 (0.37) HDAC6HDAC3HDAC4HDAC1HDAC2
SCHEMBL28579646 0.85 HDAC3 (0.35) HDAC6HDAC3HDAC4HDAC1HDAC2
SCHEMBL28915301 0.85 HDAC3 (0.36) IKBKBHDAC6HDAC3HDAC4HDAC1
SCHEMBL28588602 0.85 IKBKB (0.40) IKBKBHDAC6HDAC3HDAC4HDAC1
SCHEMBL28582707 0.84 HDAC6 (0.44) IKBKBHDAC6HDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109384793-B Thiol compound with HDAC6 inhibitory activity and application thereof 沈阳药科大学 2021-05-07 CN claimed
CN-109384793-B Thiol compound with HDAC6 inhibitory activity and application thereof 沈阳药科大学 2021-05-07 CN disclosed