SCHEMBL28600596

SCHEMBL28600596

COc1cc(Br)c[c]c1N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MAPT P10636 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
APP P05067 2/20 0.35
GAA P10253 4/20 0.34
ALDH1A1 P00352 3/20 0.34
ERN1 O75460 1/20 0.34
ALOX15 P16050 1/20 0.34
ALOX12 P18054 1/20 0.34
CYP3A4 P08684 2/20 0.33
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
MGAM O43451 1/20 0.33
SI P14410 1/20 0.33
MGAM2 Q2M2H8 1/20 0.33
NQO2 P16083 2/20 0.33
NPC1 O15118 1/20 0.32
GFER P55789 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28851924 0.78 ERN1 (0.36) POLBL3MBTL1MAPTNPSR1APP
SCHEMBL28805089 0.77 POLB (0.39) POLBL3MBTL1MAPTNPSR1APP
SCHEMBL28179999 0.77 ERN1 (0.35) POLBL3MBTL1MAPTNPSR1APP
SCHEMBL3594844 0.75 ERN1 (0.42) L3MBTL1MAPTAPPGAAALDH1A1
SCHEMBL3173111 0.75
SCHEMBL7458455 0.71
SCHEMBL1000103 0.70 MAPT (0.58) POLBL3MBTL1MAPTNPSR1APP
SCHEMBL27429619 0.70
SCHEMBL2498762 0.65 MAPT (0.52) POLBL3MBTL1MAPTNPSR1APP
SCHEMBL31211203 0.65 MAPT (0.57) POLBL3MBTL1MAPTNPSR1APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108239074-B Quinazoline compound, preparation method, application and pharmaceutical composition thereof 中国医学科学院药物研究所 2021-07-06 CN disclosed
CN-108239076-B Quinazoline compound, preparation method, application and pharmaceutical composition thereof 中国医学科学院药物研究所 2021-07-06 CN disclosed
CN-108239075-B Quinazoline compound, preparation method, application and pharmaceutical composition thereof 中国医学科学院药物研究所 2021-07-02 CN disclosed