SCHEMBL28600674

SCHEMBL28600674

Cc1cnc(Nc2cnn(C)c2)nc1-c1ccccc1C(=O)NC(C)C#N

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 10/20 0.52
JAK2 O60674 8/20 0.52
JAK3 P52333 8/20 0.50
TYK2 P29597 6/20 0.50
STAT3 P40763 3/20 0.50
FLT4 P35916 4/20 0.47
GSK3B P49841 3/20 0.47
KDR P35968 3/20 0.47
AURKB Q96GD4 3/20 0.47
ABL1 P00519 1/20 0.47
CDC7 O00311 2/20 0.44
DAPK3 O43293 2/20 0.44
ROCK2 O75116 2/20 0.44
PRKD3 O94806 2/20 0.44
MAP4K4 O95819 2/20 0.44
PAK4 O96013 2/20 0.44
PIM1 P11309 2/20 0.44
PRKACA P17612 2/20 0.44
CDK2 P24941 2/20 0.44
SYK P43405 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28605522 0.88 JAK3 (0.47) JAK1JAK2JAK3TYK2STAT3
SCHEMBL28612508 0.88 FLT4 (0.49) JAK1JAK2JAK3FLT4KDR
SCHEMBL30956392 0.86 DDR2 (0.46) JAK1JAK2JAK3TYK2FLT4
SCHEMBL28598992 0.85 IGF1R (0.54) FLT4CDK2CDK7CDK9CDK8
SCHEMBL28603799 0.84 IGF1R (0.46) JAK1JAK2JAK3FLT4KDR
SCHEMBL30956586 0.83 JAK1 (0.60) JAK1JAK2JAK3TYK2STAT3
SCHEMBL22097761 0.83 JAK2 (0.54) JAK1JAK2JAK3TYK2STAT3
SCHEMBL22089670 0.83 JAK2 (0.54) JAK1JAK2JAK3TYK2STAT3
SCHEMBL22097798 0.83 JAK2 (0.54) JAK1JAK2JAK3TYK2STAT3
SCHEMBL29942043 0.83 JAK2 (0.54) JAK1JAK2JAK3TYK2STAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113227074-A Benzamide derivatives of pyrazolyl-amino-pyrimidinyl derivatives, compositions and methods 凌科药业(杭州)有限公司 2021-08-06 CN disclosed