SCHEMBL28602196

SCHEMBL28602196

CC(C#N)NC(=O)c1ccc(-c2nc(Nc3cnn(C(C)C)c3)ncc2Cl)cc1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.44
LIMK1 P53667 1/20 0.44
AURKB Q96GD4 1/20 0.44
JAK2 O60674 11/20 0.44
JAK3 P52333 9/20 0.44
JAK1 P23458 7/20 0.44
FLT4 P35916 1/20 0.43
FLT3 P36888 6/20 0.43
TYK2 P29597 5/20 0.43
HDAC3 O15379 2/20 0.41
HDAC1 Q13547 2/20 0.41
IGF1R P08069 2/20 0.41
RPS6KB1 P23443 1/20 0.40
CDK7 P50613 1/20 0.40
CDK9 P50750 1/20 0.40
BTK Q06187 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22089934 1.00 AURKA (0.44) AURKALIMK1AURKBJAK2JAK3
SCHEMBL22098071 0.91 JAK2 (0.50) JAK2JAK3JAK1FLT3TYK2
SCHEMBL22097824 0.90 MAPK1 (0.47) AURKBJAK2JAK3JAK1FLT4
SCHEMBL29941775 0.90 MAPK1 (0.47) AURKBJAK2JAK3JAK1FLT4
SCHEMBL22097850 0.90 MAPK1 (0.47) AURKBJAK2JAK3JAK1FLT4
SCHEMBL28612309 0.90 MAPK1 (0.47) AURKBJAK2JAK3JAK1FLT4
SCHEMBL22098067 0.90 JAK2 (0.43) AURKALIMK1AURKBJAK2JAK3
SCHEMBL28603999 0.90 PAK1 (0.47) AURKALIMK1AURKBJAK2JAK3
SCHEMBL22097935 0.88 HDAC3 (0.48) AURKBJAK2JAK3JAK1FLT3
SCHEMBL29249070 0.88 HDAC3 (0.48) AURKBJAK2JAK3JAK1FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113227074-A Benzamide derivatives of pyrazolyl-amino-pyrimidinyl derivatives, compositions and methods 凌科药业(杭州)有限公司 2021-08-06 CN claimed
CN-118290403-A Benzamide derivatives of pyrazolyl-amino-pyrimidinyl and compositions and methods thereof 凌科药业(杭州)有限公司 2024-07-05 CN disclosed
CN-113227074-A Benzamide derivatives of pyrazolyl-amino-pyrimidinyl derivatives, compositions and methods 凌科药业(杭州)有限公司 2021-08-06 CN disclosed