SCHEMBL28609409

SCHEMBL28609409

O=C(Nc1ccc(-c2nc(N3CCOCC3)nc(N3CCOCC3)n2)cc1)Nc1ccc2c(c1)OCO2

nearest known ligand 0.72

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MTOR P42345 20/20 0.72
PIK3CA P42336 19/20 0.72
PIK3CG P48736 16/20 0.72
PIK3CD O00329 1/20 0.66
PIK3CB P42338 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL32179 0.84 MTOR (1.00) MTORPIK3CAPIK3CG
SCHEMBL32189 0.83 MTOR (1.00) MTORPIK3CAPIK3CG
SCHEMBL32350 0.83 PIK3CA (0.84) MTORPIK3CAPIK3CG
SCHEMBL13828917 0.83 MTOR (0.58) MTORPIK3CAPIK3CG
SCHEMBL32624 0.82 PIK3CA (0.82) MTORPIK3CAPIK3CG
SCHEMBL32400 0.82 MTOR (1.00) MTORPIK3CAPIK3CGPIK3CDPIK3CB
SCHEMBL32791 0.82 PIK3CA (1.00) MTORPIK3CAPIK3CG
SCHEMBL32467 0.82 PIK3CA (1.00) MTORPIK3CAPIK3CG
SCHEMBL32289 0.82 PIK3CA (1.00) MTORPIK3CAPIK3CG
SCHEMBL13828958 0.81 MTOR (0.58) MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113045559-B Diaryl urea PI3K alpha/mTOR double-target inhibitor and pharmaceutical composition and application thereof 贵州医科大学 2022-05-20 CN disclosed
CN-113045559-A Diaryl urea PI3K alpha/mTOR double-target inhibitor and pharmaceutical composition and application thereof 贵州医科大学 2021-06-29 CN disclosed