SCHEMBL28614224

SCHEMBL28614224

C[C@H](O)CNC[C@@H](O)[C@H](Cc1ccccc1)OC(N)=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.43
TDP1 Q9NUW8 2/20 0.43
ALDH1A1 P00352 3/20 0.40
RAB9A P51151 3/20 0.40
NPC1 O15118 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
TSHR P16473 1/20 0.40
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
CTSH P09668 1/20 0.40
CTSK P43235 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
BCHE P06276 5/20 0.39
ANPEP P15144 1/20 0.39
ERAP2 Q6P179 1/20 0.39
BACE1 P56817 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28614225 1.00 KDM4E (0.43) KDM4ETDP1ALDH1A1RAB9ANPC1
SCHEMBL28628361 1.00 KDM4E (0.43) KDM4ETDP1ALDH1A1RAB9ANPC1
SCHEMBL28614227 1.00 KDM4E (0.43) KDM4ETDP1ALDH1A1RAB9ANPC1
SCHEMBL5930124 0.92 ANPEP (0.46) KDM4EALDH1A1RAB9ANPC1MEN1
SCHEMBL5930117 0.92 ANPEP (0.46) KDM4EALDH1A1RAB9ANPC1MEN1
SCHEMBL16912773 0.92 ANPEP (0.46) KDM4EALDH1A1RAB9ANPC1MEN1
SCHEMBL8577592 0.87 F2 (0.44) BCHEANPEPBACE1
SCHEMBL8580373 0.86 BCHE (0.52) BCHEANPEPBACE1
SCHEMBL5578364 0.82 CYP3A4 (0.42) ALDH1A1RAB9ANPC1TSHRCYP1A2
SCHEMBL3356361 0.82 CYP3A4 (0.42) ALDH1A1RAB9ANPC1TSHRCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113277991-B Nitrogen heterocyclic ring amino derivative, preparation method thereof and anti-HIV-1 drug 中国医学科学院医药生物技术研究所 2022-07-12 CN disclosed
CN-113277991-A Nitrogen heterocyclic ring amino derivative, preparation method thereof and anti-HIV-1 drug 中国医学科学院医药生物技术研究所 2021-08-20 CN disclosed