SCHEMBL28619100

SCHEMBL28619100

Cc1nc2ncc(-c3nc(Nc4cc[c]cn4)ncc3F)cc2n1C(C)C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 20/20 0.49
CDK2 P24941 16/20 0.49
CDK6 Q00534 16/20 0.49
CDK1 P06493 11/20 0.49
CCNB1 P14635 8/20 0.49
CCNE1 P24864 7/20 0.49
CDK7 P50613 6/20 0.49
CDK9 P50750 6/20 0.49
CCNA2 P20248 4/20 0.49
CCND3 P30281 4/20 0.49
KDR P35968 3/20 0.49
CCNT1 O60563 2/20 0.49
EGFR P00533 2/20 0.49
NTRK1 P04629 2/20 0.49
BRAF P15056 2/20 0.49
MAPK8 P45983 2/20 0.49
CCNH P51946 2/20 0.49
MNAT1 P51948 2/20 0.49
MAPK10 P53779 2/20 0.49
CDK5 Q00535 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21955496 0.87 CDK4 (0.63) CDK4CDK2CDK6CDK1CCNB1
SCHEMBL19209867 0.78 CDK6 (0.80) CDK4CDK2CDK6CDK1CCNB1
SCHEMBL19209863 0.78 CDK6 (0.70) CDK4CDK2CDK6CDK1CCNB1
SCHEMBL19231897 0.78 CDK6 (0.61) CDK4CDK2CDK6CDK1CCNB1
SCHEMBL19231772 0.78 CDK6 (0.74) CDK4CDK2CDK6CDK1CCNB1
SCHEMBL19231823 0.78 CDK6 (0.65) CDK4CDK2CDK6CDK1CCNB1
SCHEMBL19209801 0.77 CDK6 (0.67) CDK4CDK2CDK6CDK1CCNB1
SCHEMBL19231778 0.77 CDK4 (0.80) CDK4CDK2CDK6CDK1CCNB1
SCHEMBL19231773 0.77 CDK4 (0.80) CDK4CDK2CDK6CDK1CCNB1
SCHEMBL19231763 0.77 CDK6 (0.68) CDK4CDK2CDK6CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602799-B Kinase inhibitor 上海复尚慧创医药研究有限公司 2021-08-03 CN disclosed