SCHEMBL28627693

SCHEMBL28627693

COC(=O)CNCc1ccc(-c2noc(-c3ccc(OC(C)C)c(C#N)c3)n2)cc1

nearest known ligand 0.62

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.62
S1PR3 Q99500 7/20 0.58
S1PR5 Q9H228 2/20 0.58
KCNH2 Q12809 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28926070 0.89 S1PR1 (0.59) S1PR1S1PR3S1PR5
SCHEMBL28636073 0.89 S1PR1 (0.59) S1PR1S1PR3S1PR5
SCHEMBL28633912 0.84 S1PR1 (0.59) S1PR1S1PR3
SCHEMBL6113696 0.83 S1PR1 (0.56) S1PR1S1PR3S1PR5KCNH2
Hydrochloric Acid SCHEMBL28652284 0.81 S1PR1 (0.59) S1PR1S1PR3S1PR5
Hydrochloric Acid SCHEMBL28640825 0.81 S1PR1 (0.66) S1PR1S1PR3S1PR5
Hydrochloric Acid SCHEMBL28631882 0.80 S1PR1 (0.58) S1PR1S1PR3S1PR5KCNH2
SCHEMBL28633863 0.80 S1PR1 (0.58) S1PR1S1PR3S1PR5
SCHEMBL2132920 0.80 S1PR1 (0.62) S1PR1S1PR3S1PR5KCNH2
SCHEMBL2131514 0.80 S1PR1 (0.65) S1PR1S1PR3S1PR5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109956912-B Carboxylic acid compound containing diphenyl oxadiazole, preparation method and medical application thereof 中国医学科学院药物研究所 2021-10-22 CN disclosed
CN-107827837-B Sphingosine-1-phosphate receptor modulator compounds, and preparation method and application thereof 苏州朗科生物技术股份有限公司 2021-09-24 CN disclosed