SCHEMBL28629078

SCHEMBL28629078

O=c1nc(-c2ccc(Cl)cc2)[nH]o1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.46
MAPK1 P28482 1/20 0.45
KDM4E B2RXH2 1/20 0.43
TNKS2 Q9H2K2 4/20 0.42
TNKS O95271 3/20 0.42
PARP2 Q9UGN5 2/20 0.42
GUSB P08236 1/20 0.42
ALPL P05186 2/20 0.42
DCUN1D1 Q96GG9 1/20 0.41
WNT3A P56704 1/20 0.40
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
TYMP P19971 1/20 0.39
PARP1 P09874 1/20 0.39
NR1H2 P55055 1/20 0.39
NR1H3 Q13133 1/20 0.39
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1437113 0.81 PARP1 (0.42) MAPK1KDM4ETNKS2TNKSNPC1
SCHEMBL15041027 0.81 TNKS2 (0.42) NOTUMMAPK1TNKS2TNKSDCUN1D1
SCHEMBL28669192 0.81 TNKS (0.42) NOTUMKDM4ETNKS2TNKSPARP2
SCHEMBL3743781 0.80 BTK (0.44) MAPK1KDM4ETNKS2TNKSDCUN1D1
SCHEMBL2440192 0.77
SCHEMBL28613594 0.77 ATM (0.47) NOTUMMAPK1KDM4ETNKS2TNKS
SCHEMBL7285207 0.77 KDM4E (0.47) KDM4ENPC1RAB9APARP1ALDH1A1
SCHEMBL15034646 0.77 TNKS (0.47) NOTUMKDM4ETNKS2TNKSNPC1
SCHEMBL15807126 0.77 NOTUM (0.45) NOTUMALPLNPC1RAB9ASMN1; SMN2
Hydrochloric Acid SCHEMBL9980654 0.75 HRH3 (0.42) KDM4ETNKS2TNKSNPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113735770-B Method for synthesizing 1-aminoisoquinoline skeleton by rhodium-catalyzed 4-phenyl oxadiazolone and vinylene carbonate 四川大学 2023-06-06 CN disclosed
CN-113735770-A Method for synthesizing 1-aminoisoquinoline skeleton from 4-phenyloxadiazolone and vinylene carbonate under catalysis of rhodium 四川大学 2021-12-03 CN disclosed
CN-113185537-A Rhodium-catalyzed reaction of 4-phenyloxadiazolone and vinylene carbonate for synthesizing three types of isoquinoline heterocycle 四川大学 2021-07-30 CN disclosed