SCHEMBL28630408

SCHEMBL28630408

Cc1cc(C)n(-c2cc(NC(=O)Oc3ccc(C(=O)Nc4ccccc4N)cc3)nc(-c3ccc(C)o3)n2)n1

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 19/20 0.56
ADORA1 P30542 14/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2D6 P10635 1/20 0.56
KCNH2 Q12809 3/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28630409 0.89 ADORA2A (0.71) ADORA2AADORA1CYP3A4CYP2D6KCNH2
SCHEMBL28627607 0.87 ADORA2A (0.63) ADORA2AADORA1CYP3A4CYP2D6KCNH2
SCHEMBL28623141 0.86 ADORA2A (0.69) ADORA2AADORA1CYP3A4CYP2D6KCNH2
SCHEMBL28633899 0.85 ADORA2A (0.58) ADORA2AADORA1CYP3A4CYP2D6KCNH2
SCHEMBL28636038 0.85 ADORA2A (0.57) ADORA2AADORA1CYP3A4CYP2D6KCNH2
SCHEMBL28634426 0.81 ADORA2A (0.62) ADORA2AADORA1CYP3A4CYP2D6KCNH2
SCHEMBL1490222 0.76 ADORA2A (0.73) ADORA2AADORA1CYP3A4CYP2D6KCNH2
SCHEMBL28627608 0.75 ADORA2A (0.80) ADORA2AADORA1CYP3A4CYP2D6KCNH2
SCHEMBL28636134 0.75 ADORA2A (0.64) ADORA2AADORA1CYP3A4CYP2D6KCNH2
SCHEMBL1490097 0.75 ADORA2A (0.72) ADORA2AADORA1CYP3A4CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113387938-B Substituted pyrimidine compound, preparation method, intermediate and application thereof 上海科技大学 2023-08-18 CN disclosed
CN-113387938-A Substituted pyrimidine compound, preparation method, intermediate and application thereof 上海科技大学 2021-09-14 CN disclosed