SCHEMBL28633351

SCHEMBL28633351

Nc1ccccc1NC(=O)C=Cc1ccc(CNC2CC2c2ccc(F)cc2)cc1

nearest known ligand 0.85

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 16/20 0.85
HDAC1 Q13547 6/20 0.85
MAOA P21397 4/20 0.85
HDAC2 Q92769 4/20 0.85
HDAC5 Q9UQL6 1/20 0.62
HDAC6 Q9UBN7 2/20 0.55
MAOB P27338 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29721324 1.00 KDM1A (0.85) KDM1AHDAC1MAOAHDAC2HDAC5
SCHEMBL19609272 1.00 KDM1A (0.85) KDM1AHDAC1MAOAHDAC2HDAC5
Trifluoroacetic Acid SCHEMBL29720965 0.95 KDM1A (0.80) KDM1AHDAC1MAOAHDAC2HDAC5
SCHEMBL19609273 0.86 KDM1A (0.70) KDM1AHDAC1MAOAHDAC2HDAC5
SCHEMBL19609872 0.84 KDM1A (0.83) KDM1AHDAC1MAOAHDAC2HDAC5
SCHEMBL28271443 0.81 KDM1A (0.68) KDM1AHDAC1MAOAHDAC2HDAC5
SCHEMBL1063750 0.80 HDAC1 (0.83) HDAC1HDAC2HDAC6
SCHEMBL8348757 0.80 HDAC1 (0.83) HDAC1HDAC2HDAC6
SCHEMBL1063749 0.80 HDAC1 (0.83) HDAC1HDAC2HDAC6
Trifluoroacetic Acid SCHEMBL29721116 0.79 KDM1A (0.74) KDM1AHDAC1MAOAHDAC2HDAC5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109153636-B Cyclopropyl-amide compounds as dual LSD1/HDAC inhibitors 朱比连特埃皮科尔有限责任公司 2021-10-22 CN disclosed