SCHEMBL28634428

SCHEMBL28634428

Cc1cc(C)n(-c2cc(NC(=O)COc3cccc(C(=O)NO)c3)nc(-c3ccc(C)o3)n2)n1

nearest known ligand 0.81

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 19/20 0.81
ADORA2A P29274 19/20 0.81
CYP3A4 P08684 2/20 0.77
CYP2D6 P10635 1/20 0.77
KCNH2 Q12809 1/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28627608 0.92 ADORA2A (0.80) ADORA1ADORA2ACYP3A4CYP2D6KCNH2
SCHEMBL4972610 0.88 ADORA1 (0.80) ADORA1ADORA2ACYP3A4CYP2D6KCNH2
SCHEMBL28634426 0.88 ADORA2A (0.62) ADORA1ADORA2ACYP3A4CYP2D6KCNH2
SCHEMBL4969507 0.87 ADORA2A (0.84) ADORA1ADORA2ACYP3A4CYP2D6KCNH2
SCHEMBL28636134 0.87 ADORA2A (0.64) ADORA1ADORA2ACYP3A4CYP2D6KCNH2
SCHEMBL4972664 0.87 ADORA1 (1.00) ADORA1ADORA2ACYP3A4CYP2D6KCNH2
SCHEMBL4971754 0.86 ADORA2A (1.00) ADORA1ADORA2ACYP3A4CYP2D6KCNH2
SCHEMBL4973687 0.85 ADORA1 (1.00) ADORA1ADORA2ACYP3A4CYP2D6KCNH2
SCHEMBL4973679 0.85 ADORA1 (1.00) ADORA1ADORA2ACYP3A4CYP2D6KCNH2
SCHEMBL4972636 0.84 ADORA2A (0.80) ADORA1ADORA2ACYP3A4CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113387938-A Substituted pyrimidine compound, preparation method, intermediate and application thereof 上海科技大学 2021-09-14 CN disclosed