SCHEMBL28634653

SCHEMBL28634653

COc1cc(C(=O)NCCN(C)C)c([N+](=O)[O-])cc1Nc1nccc(-c2cnn3ccccc23)n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 18/20 0.56
IGF1R P08069 2/20 0.47
INSR P06213 2/20 0.47
KCNH2 Q12809 2/20 0.47
MLNR O43193 1/20 0.44
KDM1A O60341 1/20 0.44
ABCB11 O95342 1/20 0.44
ERBB2 P04626 1/20 0.44
CHRM2 P08172 1/20 0.44
HTR1A P08908 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
DRD2 P14416 1/20 0.44
NQO2 P16083 1/20 0.44
ADRA2C P18825 1/20 0.44
DRD1 P21728 1/20 0.44
ERBB3 P21860 1/20 0.44
SLC6A2 P23975 1/20 0.44
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
ADORA2A P29274 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28637613 0.90 EGFR (0.59) EGFRIGF1RINSRKCNH2MLNR
SCHEMBL28633395 0.87 EGFR (0.56) EGFRIGF1RINSRKCNH2
SCHEMBL30219243 0.86 EGFR (0.57) EGFRIGF1RINSRKCNH2MLNR
SCHEMBL14718868 0.86 EGFR (0.57) EGFRIGF1RINSRKCNH2MLNR
SCHEMBL30883837 0.86 EGFR (0.56) EGFRIGF1RINSRKCNH2MLNR
SCHEMBL17822331 0.86 EGFR (0.56) EGFRIGF1RINSRKCNH2MLNR
SCHEMBL28628627 0.85 EGFR (0.62) EGFRIGF1RINSRKCNH2MLNR
SCHEMBL28641983 0.85 EGFR (0.66) EGFRIGF1RINSRKCNH2MLNR
SCHEMBL14663306 0.82 EGFR (0.54) EGFRIGF1R
SCHEMBL30998030 0.81 EGFR (0.55) EGFRIGF1RINSRKCNH2MLNR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107793413-B Pyrimidine heterocyclic compound and preparation method and application thereof 上海科州药物研发有限公司 2021-09-28 CN disclosed