SCHEMBL28636393

SCHEMBL28636393

COC(=O)C1CCN(Cc2ccc(-c3noc(-c4ccc(OC(C)C)c(C#N)c4)n3)cc2)C1

nearest known ligand 0.60

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 19/20 0.60
S1PR3 Q99500 6/20 0.56
MAP4K4 O95819 1/20 0.56
MINK1 Q8N4C8 1/20 0.56
S1PR5 Q9H228 2/20 0.53
S1PR4 O95977 1/20 0.53
KCNH2 Q12809 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28633782 0.92 S1PR1 (0.61) S1PR1S1PR3MAP4K4MINK1S1PR5
Hydrochloric Acid SCHEMBL28645680 0.92 MAP4K4 (0.63) S1PR1S1PR3MAP4K4MINK1S1PR5
SCHEMBL28925156 0.91 S1PR1 (0.59) S1PR1S1PR3S1PR5
SCHEMBL28632224 0.89 S1PR1 (0.54) S1PR1S1PR3MAP4K4MINK1S1PR5
SCHEMBL28633488 0.88 S1PR1 (0.60) S1PR1S1PR3MAP4K4MINK1S1PR5
SCHEMBL28926108 0.86 S1PR1 (0.64) S1PR1S1PR3MAP4K4MINK1S1PR5
SCHEMBL28631872 0.84 S1PR1 (0.58) S1PR1S1PR3MAP4K4MINK1S1PR5
SCHEMBL1967407 0.84 MAP4K4 (0.78) S1PR1S1PR3MAP4K4MINK1S1PR5
Hydrochloric Acid SCHEMBL28651669 0.84 MAP4K4 (0.61) S1PR1S1PR3MAP4K4MINK1S1PR5
Hydrochloric Acid SCHEMBL28647662 0.84 S1PR1 (0.63) S1PR1S1PR3MAP4K4MINK1S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109956912-B Carboxylic acid compound containing diphenyl oxadiazole, preparation method and medical application thereof 中国医学科学院药物研究所 2021-10-22 CN disclosed
CN-107827837-B Sphingosine-1-phosphate receptor modulator compounds, and preparation method and application thereof 苏州朗科生物技术股份有限公司 2021-09-24 CN disclosed