SCHEMBL28636876

SCHEMBL28636876

Cc1cc(Nc2ccnc(SCc3ccc(C(=O)Nc4cc(F)cc5c4=NC(=O)C=5)cc3)n2)n[nH]1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 7/20 0.49
AURKA O14965 3/20 0.42
AURKB Q96GD4 1/20 0.42
NTRK1 P04629 2/20 0.41
PKM P14618 2/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 4/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
APOBEC3A P31941 1/20 0.41
APOBEC3G Q9HC16 1/20 0.41
HDAC3 O15379 1/20 0.39
NCOR1 O75376 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23962997 0.82 HDAC1 (0.69) HDAC1AURKAAURKBNTRK1PKM
SCHEMBL23962987 0.81 HDAC1 (0.48) HDAC1AURKAAURKBNTRK1PKM
SCHEMBL23962995 0.80 HDAC1 (0.57) HDAC1AURKAAURKBNTRK1PKM
SCHEMBL23929030 0.80 HDAC1 (0.55) HDAC1AURKAAURKBNTRK1PKM
SCHEMBL23929029 0.80 HDAC1 (0.69) HDAC1AURKAAURKBPKMMAPT
SCHEMBL23929024 0.78 AURKA (0.53) HDAC1AURKAAURKBNTRK1PKM
SCHEMBL23962990 0.77 HDAC1 (0.52) HDAC1AURKAAURKBNTRK1PKM
SCHEMBL23962996 0.76 AURKA (0.52) HDAC1AURKAAURKBNTRK1SMN1; SMN2
SCHEMBL23962998 0.73 HDAC1 (0.57) HDAC1PKMMAPTNPC1RAB9A
SCHEMBL23929014 0.73 HDAC1 (0.70) HDAC1PKMMAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113549057-A Snail inhibitor and derivative thereof, preparation method, pharmaceutical composition and application 中国药科大学 2021-10-26 CN claimed
CN-113549057-B Snail inhibitor and derivative thereof, preparation method, pharmaceutical composition and application 中国药科大学 2023-01-31 CN disclosed
CN-113549057-A Snail inhibitor and derivative thereof, preparation method, pharmaceutical composition and application 中国药科大学 2021-10-26 CN disclosed