SCHEMBL28637429

SCHEMBL28637429

COCCN(C)c1ccc(C#CC(C)(O)c2nccs2)cc1Nc1ccnc2[nH]ccc12

nearest known ligand 0.81

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAP3K14 Q99558 20/20 0.81
JAK1 P23458 1/20 0.48
JAK3 P52333 1/20 0.48
TNK2 Q07912 1/20 0.48
NTRK3 Q16288 1/20 0.48
LRRK2 Q5S007 1/20 0.48
AURKB Q96GD4 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28638952 0.90 MAP3K14 (1.00) MAP3K14JAK1JAK3TNK2NTRK3
SCHEMBL30516460 0.88 MAP3K14 (0.79) MAP3K14JAK1JAK3TNK2NTRK3
SCHEMBL28639735 0.88 MAP3K14 (0.79) MAP3K14JAK1JAK3TNK2NTRK3
SCHEMBL1613463 0.78 MAP3K14 (0.68) MAP3K14
SCHEMBL1613687 0.78 MAP3K14 (0.68) MAP3K14
SCHEMBL1613461 0.78 MAP3K14 (0.68) MAP3K14
SCHEMBL30516469 0.77 MAP3K14 (0.87) MAP3K14JAK1JAK3TNK2NTRK3
SCHEMBL28657438 0.77 MAP3K14 (0.87) MAP3K14JAK1JAK3TNK2NTRK3
SCHEMBL28636846 0.77 MAP3K14 (1.00) MAP3K14JAK1JAK3TNK2NTRK3
SCHEMBL30516450 0.77 MAP3K14 (1.00) MAP3K14JAK1JAK3TNK2NTRK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112794855-B Preparation method and application of N-aryl pyrimidine-4-amine derivative 中国药科大学 2023-07-28 CN claimed
CN-112794855-A N-aryl pyrimidine-4-amine derivative and application thereof 中国药科大学 2021-05-14 CN claimed
CN-112794855-B Preparation method and application of N-aryl pyrimidine-4-amine derivative 中国药科大学 2023-07-28 CN disclosed
CN-112794855-A N-aryl pyrimidine-4-amine derivative and application thereof 中国药科大学 2021-05-14 CN disclosed