SCHEMBL28644183

SCHEMBL28644183

COC(=O)Cn1cc(-c2cccc(F)c2Cl)c(=O)n([C@@H](C)CNC(=O)OC(C)(C)C)c1=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GNRHR P30968 5/20 0.35
CYP3A4 P08684 2/20 0.34
DHODH Q02127 1/20 0.33
MALT1 Q9UDY8 1/20 0.32
UTS2R Q9UKP6 1/20 0.32
P2RX3 P56373 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
HPGD P15428 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
NCOA1 Q15788 1/20 0.32
NCOA3 Q9Y6Q9 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
KCNA5 P22460 1/20 0.32
PDPK1 O15530 1/20 0.32
CCNB2 O95067 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28644185 1.00 GNRHR (0.35) GNRHRCYP3A4DHODHMALT1UTS2R
SCHEMBL19873904 0.92 GNRHR (0.36) GNRHRCYP3A4DHODHMALT1UTS2R
SCHEMBL17870696 0.92 GNRHR (0.36) GNRHRCYP3A4DHODHMALT1UTS2R
SCHEMBL19873888 0.88 GNRHR (0.34) GNRHRCYP3A4DHODHMALT1UTS2R
SCHEMBL30178450 0.88 GNRHR (0.34) GNRHRCYP3A4DHODHMALT1UTS2R
SCHEMBL19873887 0.88 GNRHR (0.34) GNRHRCYP3A4DHODHMALT1UTS2R
SCHEMBL28644101 0.84 GNRHR (0.40) GNRHRCYP3A4P2RX3SMN1; SMN2KDM4E
SCHEMBL28641621 0.84 GNRHR (0.39) GNRHRCYP3A4P2RX3KDM4EALDH1A1
SCHEMBL28663476 0.84 GNRHR (0.39) GNRHRCYP3A4P2RX3KDM4EMEN1
SCHEMBL28663474 0.84 GNRHR (0.39) GNRHRCYP3A4P2RX3KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107428744-B Novel heterocyclic compounds and their use in medicine and cosmetics 盖尔德马研究及发展公司 2021-09-24 CN disclosed