SCHEMBL28645932

SCHEMBL28645932

Cc1nc(Nc2n[nH]c3c2CN(C(=O)O)C3(C)C)c2ccsc2n1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PAK4 O96013 18/20 0.71
OPRM1 P35372 1/20 0.53
PRKCB P05771 3/20 0.52
PLK4 O00444 1/20 0.52
CHEK1 O14757 1/20 0.52
AURKA O14965 1/20 0.52
GAK O14976 1/20 0.52
RPS6KA5 O75582 1/20 0.52
RPS6KA4 O75676 1/20 0.52
STK16 O75716 1/20 0.52
PAK3 O75914 1/20 0.52
CDKL5 O76039 1/20 0.52
PRKD3 O94806 1/20 0.52
LATS1 O95835 1/20 0.52
CHEK2 O96017 1/20 0.52
NTRK1 P04629 1/20 0.52
TP53 P04637 1/20 0.52
PRKCG P05129 1/20 0.52
FYN P06241 1/20 0.52
YES1 P07947 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22164663 0.87 PAK4 (0.66) PAK4OPRM1PRKCBPLK4CHEK1
SCHEMBL29412167 0.84 PAK4 (0.65) PAK4OPRM1PRKCBPLK4CHEK1
SCHEMBL1942289 0.84 PAK4 (1.00) PAK4OPRM1
SCHEMBL1369727 0.84 PAK4 (1.00) PAK4OPRM1
SCHEMBL1369729 0.84 PAK4 (1.00) PAK4OPRM1
SCHEMBL1942571 0.82 PAK4 (0.80) PAK4PRKCBPLK4CHEK1AURKA
SCHEMBL1941057 0.81 PAK4 (1.00) PAK4PRKCBPLK4CHEK1AURKA
SCHEMBL3503797 0.81 PAK4 (1.00) PAK4PRKCBPLK4CHEK1AURKA
SCHEMBL1941053 0.80 PAK4 (0.71) PAK4OPRM1PRKCBPLK4CHEK1
SCHEMBL1941054 0.79 PAK4 (0.66) PAK4OPRM1PRKCBPLK4CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113557017-A Inhibitors of cyclin-dependent kinase 7 and uses thereof 达纳-法伯癌症研究所股份有限公司 2021-10-26 CN disclosed