SCHEMBL28650052

SCHEMBL28650052

O=[N+]([O-])c1c(Cl)ncnc1N1CCOCC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CUL4A Q13619 1/20 0.49
CYP1A2 P05177 4/20 0.49
CYP2C9 P11712 4/20 0.49
RPS6KB1 P23443 2/20 0.46
KDM4E B2RXH2 1/20 0.45
GAA P10253 1/20 0.45
ALDH1A1 P00352 5/20 0.45
POLB P06746 1/20 0.43
HPGD P15428 1/20 0.43
MAPT P10636 5/20 0.43
CYP2C19 P33261 2/20 0.43
CYP3A4 P08684 1/20 0.43
PTK2 Q05397 1/20 0.42
MGMT P16455 1/20 0.42
MAPK1 P28482 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HTT P42858 1/20 0.41
CHEK1 O14757 1/20 0.41
PDPK1 O15530 1/20 0.41
PAK1 Q13153 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30623370 1.00 CUL4A (0.49) CUL4ACYP1A2CYP2C9RPS6KB1KDM4E
SCHEMBL30623376 0.86 CUL4A (0.59) CUL4ACYP1A2CYP2C9RPS6KB1ALDH1A1
SCHEMBL28644797 0.86 CUL4A (0.59) CUL4ACYP1A2CYP2C9RPS6KB1ALDH1A1
SCHEMBL30623383 0.85 CUL4A (0.57) CUL4ACYP1A2CYP2C9RPS6KB1ALDH1A1
SCHEMBL28650731 0.85 CUL4A (0.57) CUL4ACYP1A2CYP2C9RPS6KB1ALDH1A1
SCHEMBL12604551 0.81 CUL4A (0.48) CUL4ACYP1A2CYP2C9RPS6KB1CYP2C19
SCHEMBL3435512 0.80 CUL4A (0.53) CUL4ARPS6KB1ALDH1A1POLBHPGD
SCHEMBL6948779 0.79 HTT (0.52) CUL4ACYP1A2CYP2C9RPS6KB1KDM4E
SCHEMBL28648550 0.78 CUL4A (0.51) CUL4AMAPK1NPSR1HTT
SCHEMBL30623361 0.78 CUL4A (0.51) CUL4AMAPK1NPSR1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113620976-B Thiazolopyrimidine compound, preparation method, application and pharmaceutical composition thereof 中国医学科学院药物研究所 2023-09-26 CN disclosed
CN-113620976-A Thiazolopyrimidine compound and preparation method, application and pharmaceutical composition thereof 中国医学科学院药物研究所 2021-11-09 CN disclosed