SCHEMBL28650246

SCHEMBL28650246

COc1cc2c(c(F)c1Br)OC[C@H]1CN(C(=O)O)CCN1C2=O

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KRAS P01116 4/20 0.47
DPP4 P27487 1/20 0.33
KDM4E B2RXH2 2/20 0.33
CYP3A4 P08684 1/20 0.33
PKM P14618 1/20 0.33
TSHR P16473 1/20 0.33
KCNJ1 P48048 3/20 0.32
ALDH1A1 P00352 1/20 0.32
HTR2A P28223 2/20 0.32
HTR2C P28335 2/20 0.32
HTR2B P41595 2/20 0.32
KMT2A Q03164 1/20 0.32
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
ALPL P05186 2/20 0.31
MGLL Q99685 1/20 0.31
MAPT P10636 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28650919 0.90 KRAS (0.42) KRASDPP4MGLL
SCHEMBL28674435 0.88 KRAS (0.43) KRASHTR2AHTR2CHTR2BALPL
SCHEMBL24558469 0.88 KRAS (0.44) KRAS
SCHEMBL29693097 0.88 KRAS (0.44) KRAS
SCHEMBL28658815 0.88 KRAS (0.41) KRASDPP4
SCHEMBL28929459 0.86 KRAS (0.44) KRASDPP4
SCHEMBL28651201 0.85 KRAS (0.45) KRASDPP4
SCHEMBL28671505 0.85 KRAS (0.40) KRASDPP4
SCHEMBL24558322 0.80 KRAS (0.41) KRASDPP4
SCHEMBL28674439 0.80 KRAS (0.40) KRASDPP4MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113508118-A Fused tricyclic compounds useful as anticancer agents 阿斯利康(瑞典)有限公司 2021-10-15 CN disclosed