SCHEMBL28656185

SCHEMBL28656185

Cc1cccc(-c2noc(-c3ccc(I)c(O)c3)n2)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 5/20 0.45
NPC1 O15118 10/20 0.43
RAB9A P51151 10/20 0.43
TP53 P04637 8/20 0.43
MAPT P10636 8/20 0.43
PKM P14618 7/20 0.43
TSHR P16473 5/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
S1PR1 P21453 2/20 0.42
SMN1; SMN2 Q16637 8/20 0.41
HSD17B10 Q99714 4/20 0.41
KDM4E B2RXH2 3/20 0.41
NPSR1 Q6W5P4 2/20 0.41
ALDH1A1 P00352 2/20 0.41
LMNA P02545 2/20 0.41
KLF5 Q13887 2/20 0.41
MAPK1 P28482 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MITF O75030 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28653851 0.87 S1PR1 (0.55) GRM5NPC1RAB9ATP53MAPT
SCHEMBL28659798 0.86 GRM5 (0.46) GRM5NPC1RAB9ATP53MAPT
SCHEMBL28665260 0.85 NPC1 (0.51) GRM5NPC1RAB9ATP53MAPT
SCHEMBL28661994 0.85 GRM5 (0.45) GRM5NPC1RAB9ATP53MAPT
SCHEMBL28654922 0.82 NPC1 (0.54) GRM5NPC1RAB9ATP53MAPT
SCHEMBL28664806 0.81 GRM5 (0.52) GRM5NPC1RAB9ATP53MAPT
SCHEMBL28656184 0.78 S1PR1 (0.48) NPC1RAB9ATP53MAPTS1PR1
SCHEMBL20968286 0.72 SMN1; SMN2 (0.52) NPC1RAB9ATP53MAPTPKM
SCHEMBL8000260 0.66 SNCA (0.55) NPC1RAB9ATP53MAPTTSHR
SCHEMBL26693406 0.66 USP7 (0.41) NPC1RAB9AS1PR1KDM4EL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113603684-B 1,2, 4-oxadiazole Nrf2 activator-tac Lin Pinge product and preparation method and application thereof 中国药科大学 2023-12-19 CN disclosed
CN-113603684-A 1,2, 4-oxadiazole Nrf2 activator-tacrine split product and preparation method and application thereof 中国药科大学 2021-11-05 CN disclosed