SCHEMBL28660573

SCHEMBL28660573

c1ccc(COC2CNC2)nc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.56
MGMT P16455 1/20 0.46
DRD4 P21917 1/20 0.44
SIGMAR1 Q99720 1/20 0.44
SYK P43405 2/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CASP6 P55212 1/20 0.39
AURKB Q96GD4 1/20 0.39
INCENP Q9NQS7 1/20 0.39
HRH1 P35367 1/20 0.39
NPC1 O15118 1/20 0.39
LMNA P02545 1/20 0.39
RAB9A P51151 1/20 0.39
ABCB1 P08183 1/20 0.39
HTR1A P08908 1/20 0.39
DRD2 P14416 1/20 0.39
PARP10 Q53GL7 1/20 0.39
LPL P06858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25258863 0.87 CHRM2 (0.54) SLC6A4MGMTDRD4SIGMAR1
SCHEMBL12120447 0.87 CHRM2 (0.54) SLC6A4MGMTDRD4SIGMAR1
SCHEMBL25258864 0.87 CHRM2 (0.54) SLC6A4MGMTDRD4SIGMAR1
Hydrochloric Acid SCHEMBL31400380 0.86 CHRM2 (0.52) SLC6A4MGMTDRD4SIGMAR1
SCHEMBL1001296 0.85 CHRM2 (0.58) SLC6A4MGMTDRD4SIGMAR1ALDH1A1
SCHEMBL8310750 0.83 SLC6A4 (0.50) SLC6A4MGMTDRD4SIGMAR1ALDH1A1
SCHEMBL15477305 0.81 DRD4 (0.51) SLC6A4MGMTDRD4SIGMAR1SYK
SCHEMBL3920378 0.78 DRD4 (0.49) SLC6A4MGMTDRD4SIGMAR1SYK
Hydrochloric Acid SCHEMBL7924437 0.76 SLC6A4 (0.42) SLC6A4MGMTDRD4SIGMAR1SYK
SCHEMBL536843 0.74 DRD4 (0.44) SLC6A4MGMTDRD4SIGMAR1SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110177786-B Substituted pyrazolo [1,5-A ] pyridine compounds as RET kinase inhibitors 阿雷生物药品公司 2021-12-14 CN disclosed