SCHEMBL28672102

SCHEMBL28672102

CC(C)(C)C1C(c2cc3cn[nH]c3c(-c3ccc(Oc4ccccc4)cc3)n2)CCN1C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BTK Q06187 17/20 0.57
EGFR P00533 1/20 0.36
TEC P42680 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CPT2 P23786 1/20 0.34
CPT1A P50416 1/20 0.34
MCL1 Q07820 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28689145 0.82 BTK (0.61) BTKMEN1KMT2A
SCHEMBL20572741 0.79 BTK (0.61) BTKCPT2CPT1A
SCHEMBL16597622 0.79 BTK (0.56) BTKEGFRTEC
SCHEMBL19203181 0.76 BTK (0.70) BTK
SCHEMBL19202621 0.75 BTK (0.59) BTKEGFRTEC
SCHEMBL19202386 0.74 BTK (0.70) BTKEGFRTEC
SCHEMBL19202347 0.74 BTK (0.70) BTKEGFRTEC
SCHEMBL19202381 0.74 BTK (0.70) BTKEGFRTEC
SCHEMBL20573086 0.74 BTK (0.74) BTK
SCHEMBL17983499 0.74 BTK (0.44) BTKEGFRTEC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602818-B Pyrazole fused ring derivatives, preparation method thereof and application thereof in treating cancer, inflammation and immune diseases 北京诺诚健华医药科技有限公司 2021-12-21 CN disclosed