SCHEMBL28680996

SCHEMBL28680996

CCNC(=O)NS(=O)(=O)c1cnccc1Nc1cccc(C)c1

nearest known ligand 0.79

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 5/20 0.74
KDM4E B2RXH2 1/20 0.74
CYP3A4 P08684 1/20 0.74
CYP2C9 P11712 1/20 0.74
HIF1A Q16665 1/20 0.74
PTGS1 P23219 3/20 0.53
PTGS2 P35354 2/20 0.53
PIK3CA P42336 1/20 0.45
MAPK8 P45983 1/20 0.45
MAPK9 P45984 1/20 0.45
MAPK10 P53779 1/20 0.45
BRS3 P32247 2/20 0.44
NAMPT P43490 2/20 0.43
PKM P14618 1/20 0.43
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29833136 1.00 TBXA2R (0.74) TBXA2RKDM4ECYP3A4CYP2C9HIF1A
SCHEMBL5668299 0.92 TBXA2R (0.71) TBXA2RKDM4ECYP3A4CYP2C9HIF1A
SCHEMBL28655173 0.90 TBXA2R (0.69) TBXA2RKDM4ECYP3A4CYP2C9HIF1A
SCHEMBL29832825 0.90 TBXA2R (0.69) TBXA2RKDM4ECYP3A4CYP2C9HIF1A
SCHEMBL13284096 0.86 TBXA2R (0.81) TBXA2RKDM4ECYP3A4CYP2C9HIF1A
Torsemide SCHEMBL5434259 0.86 TBXA2R (0.92) TBXA2RKDM4ECYP3A4CYP2C9HIF1A
Torsemide SCHEMBL4015063 0.85 TBXA2R (1.00) TBXA2RKDM4ECYP3A4CYP2C9HIF1A
Torsemide SCHEMBL41184 0.85 TBXA2R (1.00) TBXA2RKDM4ECYP3A4CYP2C9HIF1A
SCHEMBL32688080 0.85 TBXA2R (0.68) TBXA2RKDM4ECYP3A4CYP2C9HIF1A
Torsemide SCHEMBL29369134 0.85 TBXA2R (1.00) TBXA2RKDM4ECYP3A4CYP2C9HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115010659-A New impurity reference substance of torasemide and preparation method thereof 南京正科医药股份有限公司 2022-09-06 CN disclosed
CN-114989077-A New impurity reference substance of torasemide and synthetic method thereof 南京正科医药股份有限公司 2022-09-02 CN disclosed
CN-113620868-A Torasemide new impurity and preparation method thereof 南京恒正药物研究院有限公司 2021-11-09 CN disclosed