SCHEMBL28686135

SCHEMBL28686135

CCOC(=O)c1[nH]nc2c1CNC(C)C2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.40
MAPK10 P53779 1/20 0.40
RIPK1 Q13546 1/20 0.40
HSD17B10 Q99714 3/20 0.39
PDE4D Q08499 1/20 0.38
MAPT P10636 2/20 0.36
KDM4E B2RXH2 5/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 4/20 0.35
ALDH1A1 P00352 2/20 0.35
HTT P42858 1/20 0.35
RECQL P46063 1/20 0.35
BRD4 O60885 1/20 0.34
ALOX15 P16050 1/20 0.34
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
CDC25B P30305 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22746962 1.00 AURKA (0.40) AURKAMAPK10RIPK1HSD17B10PDE4D
Hydrochloric Acid SCHEMBL29071885 0.99 AURKA (0.40) AURKAMAPK10RIPK1HSD17B10PDE4D
Hydrochloric Acid SCHEMBL29071888 0.99 AURKA (0.40) AURKAMAPK10RIPK1HSD17B10PDE4D
SCHEMBL23513289 0.83 BRD4 (0.42) MAPTLMNAALDH1A1BRD4POLB
SCHEMBL22717992 0.80 HCAR2 (0.35) HSD17B10KDM4EALDH1A1
SCHEMBL22717989 0.80 HCAR2 (0.35) HSD17B10KDM4EALDH1A1
SCHEMBL19140474 0.76 KDM4E (0.45) AURKAMAPK10RIPK1HSD17B10PDE4D
SCHEMBL23513389 0.75 AURKA (0.44) AURKAMAPK10RIPK1HSD17B10PDE4D
SCHEMBL30092714 0.75 AURKA (0.40) AURKAMAPK10RIPK1HSD17B10PDE4D
SCHEMBL29515403 0.74 SMN1; SMN2 (0.39) AURKAMAPK10RIPK1HSD17B10PDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117715909-A Condensed heterocyclic derivative 杨森科学爱尔兰无限公司 2024-03-15 CN disclosed
CN-113906028-A Fused heterocyclic derivatives 爱尔兰詹森科学公司 2022-01-07 CN disclosed