SCHEMBL28688451

SCHEMBL28688451

O=C(O)c1nn(-c2ccccc2)ccc1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 1.00
KMT2A Q03164 4/20 0.73
MEN1 O00255 1/20 0.70
GAA P10253 1/20 0.69
POLB P06746 2/20 0.58
MAPK1 P28482 1/20 0.51
ALDH1A1 P00352 4/20 0.51
L3MBTL1 Q9Y468 2/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
KDM4E B2RXH2 1/20 0.50
HTT P42858 2/20 0.49
TSHR P16473 2/20 0.49
MAPT P10636 1/20 0.49
HSD17B10 Q99714 1/20 0.49
HPGD P15428 1/20 0.47
UBE2N P61088 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31261492 0.86 CYP2C9 (0.76) CYP2C9KMT2AMEN1GAAPOLB
SCHEMBL29826882 0.86 CYP2C9 (0.76) CYP2C9KMT2AMEN1GAAPOLB
SCHEMBL28662399 0.86 CYP2C9 (0.76) CYP2C9KMT2AMEN1GAAPOLB
SCHEMBL2221815 0.85 CYP2C9 (0.73) CYP2C9KMT2AMEN1GAAPOLB
SCHEMBL359785 0.83 KMT2A (0.71) CYP2C9KMT2AMEN1GAAPOLB
SCHEMBL31054400 0.81 CYP2C9 (0.69) CYP2C9KMT2AMEN1GAAPOLB
SCHEMBL518604 0.81 KMT2A (0.67) CYP2C9KMT2AMEN1GAAPOLB
SCHEMBL11397324 0.79 GAA (0.72) CYP2C9KMT2AMEN1GAAPOLB
SCHEMBL2221528 0.79 CYP2C9 (0.63) CYP2C9KMT2AMEN1GAAPOLB
SCHEMBL9594109 0.78 CYP2C9 (0.64) CYP2C9KMT2AMEN1GAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113620873-B Preparation method and application of zinc-containing binding group and quinoline skeleton compound 沈阳药科大学 2023-12-08 CN disclosed
CN-110467616-B Preparation and application of triazolopyrazine compound containing heteroaryl substituted pyridazinone structure 江西科技师范大学 2021-12-21 CN disclosed
CN-113620873-A Preparation method and application of compound containing zinc binding group and quinoline skeleton 沈阳药科大学 2021-11-09 CN disclosed