SCHEMBL28699433

SCHEMBL28699433

O=C(O)c1ccc2[nH]c(CC3CCNCC3)nc2c1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 3/20 0.53
NPSR1 Q6W5P4 1/20 0.48
HTR2B P41595 1/20 0.47
IDO1 P14902 4/20 0.46
APEX1 P27695 1/20 0.46
TOP2A P11388 1/20 0.43
KDM4E B2RXH2 1/20 0.42
RECQL P46063 1/20 0.42
CACNA1G O43497 2/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPK1 P28482 1/20 0.42
GRIN2B Q13224 1/20 0.42
CYP1A2 P05177 1/20 0.41
TSHR P16473 1/20 0.41
CHEK2 O96017 1/20 0.40
MELK Q14680 1/20 0.40
ABL1 P00519 1/20 0.39
KDM1A O60341 1/20 0.39
LGALS8 O00214 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28681429 0.83 CACNA1H (0.47) CACNA1HNPSR1KDM4EALDH1A1MAPK1
SCHEMBL29491599 0.81 NPSR1 (0.47) NPSR1HTR2BIDO1APEX1TOP2A
SCHEMBL11887806 0.79 APEX1 (0.64) NPSR1APEX1TOP2AKDM4ERECQL
Cadaverine Tartrate SCHEMBL7964690 0.79 CACNA1H (0.50) CACNA1HHTR2BIDO1CACNA1GGRIN2B
SCHEMBL4785390 0.78 NPSR1 (0.75) NPSR1APEX1TOP2AKDM4ERECQL
SCHEMBL2996556 0.76 NPSR1 (0.56) NPSR1APEX1TOP2AKDM4ERECQL
SCHEMBL29424865 0.76 NPSR1 (0.56) NPSR1APEX1TOP2AKDM4ERECQL
SCHEMBL6092621 0.76 KDM4E (0.68) NPSR1APEX1TOP2AKDM4ERECQL
Hydrochloric Acid SCHEMBL28877037 0.75 KDM4E (0.66) NPSR1APEX1TOP2AKDM4ERECQL
SCHEMBL31695078 0.75 APEX1 (0.59) NPSR1APEX1TOP2AKDM4ERECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113227068-A GLP-1R agonists and uses thereof 上海齐鲁锐格医药研发有限公司 2021-08-06 CN disclosed